Caafimaadka, Diyaarinta
The daroogada "Betagestin" ka vertigo. "Betahistine": tilmaamaha loo isticmaalo, qiimaha, dib u eegista
ma daroogada "Betahistine" (kiniin) Sidee? Tilmaamaha loogu isticmaalo, dib u eegista, sharaxaada iyo sifooyinka daroogada waxaa lagu hoos lagu soo bandhigay. Intaa waxaa dheer, waxaan kuu sheegi doonaa waxa ku saabsan qalab ay u xilsaarantahay, qiime intee le'eg, haddii ay waxyeelo kasta oo dhinaca iyo sababo.
Halabuurka, description qaabka iyo
foomka Release of daroogada ka mid ah - kaniiniga. Si kastaba ha ahaatee, la heli karo qiyaas oo ah walaxda firfircoon kala duwan:
- Valium kiniinada cadcad ee qaab wareeg ah ku tilmaamay qiyaasood oo firfircoon (dihydrochloride betahistine) - 8 mg.
- kiniin kiish oo biconvex la qaadasho fekrado geesaha ku tilmaamay ee firfircoon (dihydrochloride betahistine) - 16 ama 24 mg.
Sida maaddooyinka kaabayaal xogta qaab ka kooban sodium sulfate lauryl, sodium croscarmellose, cellulose mikrokristallin, milmahayn magnesium iyo qaarna.
tallaabada pharmacological daroogada
Waa maxay daawada "Betahistine?" Tilmaamaha loogu isticmaalo (qiimaha daawooyinka hoos ku taxan) ayaa sheegay in daroogada waa analoogga ah histamine, kaas oo lagu abuuray synthetically.
kiniiniyada awood u firfircoon ku lug H-3 histamine iyo H-1 receptors (xoog leh oo ku Doodeen daciif ah) habdhiska dhimirka (i.e., receptors ka mid ah nuclei vestibular iyo dhegaha hoose).
Ka dib markii daawada waa si degdeg ah u saameeyaa socodka dhiigga, kor u qaadida kicinta ee microcirculation iyo permeability ee qalintaanka dhegta gudaha. Sidoo kale, qayb firfircoon ee medicament waa ay awoodaan in ay xasilin cadaadiska gudaha cochlea endolymph ah.
Sababo la xaqiiqada ah in "Betahistine" waa inhibitor ah ee H 3 receptors nuclei nidaamka vestibular, waxa uu saameyn ku fahmayaan on yimaada habdhiska dhimirka. Sayidka, daroogada loo arkaa degto gudbinta (neuronal) neurons in xuduntii vestibular.
Iyada oo qiyaasta saxda ah ee daawada, inuu awoodo inuu si deg deg ah oo ku filan in la baabi'iyo Aayaadka vertigo vestibular. Time-gaadhista ee qayb firfircoon ee daroogada u dhaxeysa dhowr daqiiqo illaa hal maalin.
qaadashada joogtada ah ee daroogada iyada oo ay kormeerayaan dhakhtar yaraynaysaa dhacdooyinka wareer, yaraynaysaa wacaya iyo soo wacayo in dhegaha, iyo dib u soo celisa dhageysiga in ay sii xumaato.
daawo waxa uu leeyahay suuxin lahayn oo aanu ka dhigi rabshooyin in isuduwidda ah.
guryaha pharmacokinetic
"Betagestin" Drug ka vertigo si degdeg ah oo si buuxda u nuugo. Its uruureen dhiig peak waxaa lagu gaaraa in ku saabsan 65 daqiiqo ka dib markii soonka.
walaxda firfircoon ee medicament la xiriira protein ah in ka yar 5%.
Dheefay by daroogada metabolize in metabolites firfircoonayn - demetilbetagistina iyo 2-pyridylacetic acid. The reebay gebi ahaanba daroogada qaadataa meel inta lagu jiro maalinta iyada oo kelyaha (90%). Wixii ka haray 10%, ay soo bandhigay by xiidmaha.
Tilmaamayaasha
"Betagestin" Drug ka wareer bukaan loo xilsaaray marar aad u badan. Intaa waxaa dheer, daroogada loo isticmaalo daweynta ee Meniere ee syndrome, iyo sidoo kale in la baabi'iyo buuq dhagahiisa, lalabo, lumista maqalka ee qayb ahaan iyo isku si daciif ah.
Waa in la ogaadaa in Meniere ee syndrome teedu sida xanuunada maqalka iyo vestibular in hore aan lagu arkay bini'aadanka. Waxa kale oo dhici kara in qaab stroke ba'an. Meniere ee syndrome ayaa itimaalka sare ah soo noqoshada soo noqnoqda.
sababo
Hadda waxaad ogaan ujeedada daroogada loo isticmaalo "Betagestin". From vertigo u badbaadiyay si aad u wanaagsan. Si kastaba ha ahaatee, daroogada this waxaa jira sababo. Waa in aan qoro dadka qaba pheochromocytoma.
Tan iyo daroogada firfircoon waa analoogga ah synthetic histamine, isticmaalkeeda waxaa laga yaabaa in ay gacan sii daayo catecholamines, taas oo keenta in hypertension daran.
Sidoo kale waa in la ogaadaa in qalab ah ee Kiniinka "betahistine" yihiin in bukaanka qaba diidmo qayb firfircoon, ama wax kasta oo excipients kale ee halabuurka ah ee daroogada.
tilmaamaha daroogada
"Betagestin" Drug ka vertigo waa in la qaato si adag iyadoo la raacayo tilmaamaha la baxshay.
- Qiyaasta dadka bukaanka ah ee dadka waaweyn.
kiniiniyada "Betahistine" maamula at qiyaasta a of 8 ama 16 mg saddex jeer maalintii (bilowga ah ee daaweynta) wada jir ah ula cuntada ama ka dib. dose dayactirka The kala duwan daawo 24-48 mg maalintii (ikhtiyaar dhakhtarka).
qiyaasta maalin walba ah ee daroogada waa in aanay noqon ka badan 48 mg. Waxaa la saxo bukaanka qofka oo dhan. Mararka qaarkood horumar ah ee uu xaalad laga dheehan karo oo keliya dhowr toddobaad ka dib.
- Daaweynta dadka qaba wadnaha, kelyaha iyo beerka.
Waayo, dadka qaba cudurka sida daroogada "Betahistine" waxaa laga yaabaa in loo magacaabo oo keliya ka dib markii baaritaan caafimaad.
- Daawaynta dadka waayeelka ah.
In da 'weyn, daawada la qoray si taxadar leh u daran. Tan waxa u sabab xaqiiqada ah in kooxdan oo ah bukaan jirto suurtagalnimada weyn oo waxyeelo ka shaqeeyo in walxaha kaabayaal ah oo firfircoon, taas oo ay qayb ka yihiin Alwaaxdii.
- Daaweynta carruurta iyo dhallinyarada.
"Betagestin" Drug ka vertigo aan qoray in carruurta iyo dhallinyarada (ka yar 18 sano). Tan waxa u sabab la'aan quseeya ammaanka iyo daawooyinka xogta.
xaaladood oo badinta
Haddii xad dhaafka "Betahistine" bukaanada qaar ka mid ah la kulmi karaan calaamadaha sida lallabo, madax- xanuun, xanuun ee caloosha iyo hurdo (inta aad qaadanaysid qiyaasta kor u ah in ay 640 mg).
Sidoo kale, bukaanka waxaa laga yaabaa in ay ka cawdaan xanuun, matag, dyspepsia, iyo ataxia.
Waayo, dhibaatooyinka ka sii daran waxaa ka mid ah dhibaatooyinka wadnaha iyo sambabada (arkay la iska badiyo ula kac ah).
Daaweynta - dhaqaya caloosha 60 daqiiqo ka dib markii maamulka gudahood.
waxyeellooyin
Ma aha oo dhan bukaanka qaadanaya daawada "Betagestin", la kulmi kartaa raaxo.
Dhakhaatiirta ayaa sheegay in muujinta dhibaato marka la qaadanayo wax daawo ah bukaanka macnaheedu noqon kartaa qabsado dawooyinka cusub. In xiriir this, hubi inaad la tashato dhakhtarkaaga hor inta aysan joojin daroogada.
Waxyeelooyinka ugu badan waxa ka qaadato "betahistine" lagu arkay mid ka mid ah toban bukaan ah. Liiska saamaynta ugu badan ka soo gaartey waxaa ka mid ah calaamadaha sida:
- calool kacsan (sida caadiga ah dhacdaa marka la qaadanayo dawada cuntada ka hor);
- qidmeyntiibulshada ee guud;
- raaxo la'aan ama dibiro,
- madax xanuun (oo aad qaadi karto xanuun joojiyaha, laakiin kaliya ka dib markii la tashanaya ka hor inta aan la takhasus gaar ah);
- cadaanyo on maqaarka ee foomka of cuncun iyo finan (waa in ay qaadaan goobaha xasaasiyadda ama dufan dhibaato tire).
Haddii tilmaamaha kor ku xusan ma caawin baabi'iyo waxyeellooyinka, bukaanka u baahan yahay in uu arko dhakhtar.
Qiimaha daroogada
Price Kiniiniga "Betahistine" waxaa laga yaabaa kala duwan oo ku xiran cadadka daawada ee xirmadan. Daawada at dose oo ah 24 mg laga iibsan karaa 60-65 rubles. Bukaan badan ayaa waxay aaminsan yihiin in ay tahay arrin daroogada kharash yar.
Reviews of daawo
Reviews of "Betahistine" dejinta waa isku dhafan. Qaar ka mid ah bukaannada qaba cudurrada wadnaha chronic si joogto ah u qaadanayso kiniinnada. Si kastaba ha ahaatee, waxay had iyo jeer ma la baabi'iyo ka madax xanuun iyo wareer.
Iyo dib u eegid xun ama fiican oo ku saabsan medicament this ayaa tilmaamaya in ay u baahan tahay codsi gaar ah.
Sidaas darteed, markii mid ka mid ah xadgudubyada "Betahistine" daroogada si deg deg ah loo soo celiyo kartaa caafimaadka qofka bukaanka ah, halka ka kale, on lid ku ah, ma laha saamayn la doonayo, laakiin yareeyo kaliya muuqaalka kore ee calaamadaha.
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