Caafimaadka, Diyaarinta
"Formetin": tilmaamaha loo isticmaalo, dhabta ah
Currently waxaan ka helay dad badan oo qaba sonkorowga iyo dhibaatooyinka noocan ah cayilka. daawooyin badan oo diyaar u ah daaweynta xanuunnada kuwan. Mid ka mid ah iyaga ka mid ah waa daawo "Formetin". Its muuqaalada socodyada waa la sharaxi doonaa in this article.
category dawooyinka
"Formetin" tilmaamaha loo isticmaalo kaas oo lagu muujiyay in this article, waa koox daroogada hypoglycemic a biguanide.
Description of qaab Halabuurka iyo sii daayo
In mid ka mid ah kiniin:
m, g | m, g | m, g | |
Walaxda firfircoon | |||
hydrochloride metformin | 0.500 | 0.850 | 1000 |
walxaha kaabayaal | |||
nooca kelli dhexe povidone | 0.017 | 0.029 | 0.034 |
sodium croscarmellose | 0.008 | 0,0136 | 0.016 |
milmahayn magnesium | 0.005 | 0,0084 | 0.010 |
daroogada Available "Formetin" ee finan 100, 60 ama 30 kiniin.
Color White kiniiniyada iyo qiyaasta foomka ku xiran tahay waxyaabaha salka. At 500 mg ploskotsilindricheskoy ay leeyihiin qaab wareeg ah iyadoo la sumaddii iyo chamfered. Sidoo kale qiyaasta of 1000 mg ama 850 mg leeyahay "Formetin". The oo kiniin ah in ay taasi dhacdo, convex iyo gadood. Waxay yihiin halis hal dhinac.
pharmacodynamics
Metformin ( "Formetin") gaabisaa gluconeogenesis dal ee beerka, iyo sidaas waxaa jira hoos u dhac in waxa dukaamada glycogen. Qalabkani waxa uu ku kordhinaya dhibaatada ee nuugista ka glucose xiidmaha, kor u qaadidda heerka sonkorta dhiigga ee nidaamka. Tani waxay kordhisaa jawaabta ee unugyada in insulin la'aan saamaynaya wax soo saarka ee qayb hormoonada ay ka mid ah beeryarada B-unugyada, Goldogob reaction hypoglycemic, tan iyo markii aan la shaqeysiin saarka walax yiri.
Drug dib u eegista "Formetin" kaas oo ay ka hadlaan oo ay wax ku oolnimada, yaraynaysaa qadarka dhiigga ee kolestaroolka "xun" iyo triglycerides. content ee Lipoproteins cufnaanta sare this kordhisaa in 20-30%. Iyada oo waxtardarradoodu ee daroogada cunto tilmaamaha "Formetin" loo isticmaalo kaas oo lagu qeexay qodobka this ka caawisaa si loo yareeyo ama / iyo xasilinta miisaanka bukaanka. Tani waxay dhacdaa ay sabab u tahay qayilo ee glucose by oxygen-lacag la'aan ah iyo in la yareeyo cunto xumo. Sidoo kale waxa uu helaba unugyada geedi socodka ay hawshooda u plasminogen by simaha ay inhibitor, kuna waari dhexdeeda saamayn hemostatic u muuqdo.
Pharmacokinetics
metformin milmaan bilaabmaa mareenka caloosha iyo mindhicirka. tirada ugu badan oo ah walaxda in dhiig baa ku saabsan 2.5 saacadood ka dib codsiga at heerka of dose unit nuugista - 50-60%. tayada nuugid ee daroogada ah ee jirka ku saameeyaa xidhiidhka ka dhexeeya walaxda firfircoon iyo protein ee plasma ah. In kiniin "Formetina" xidhiidh lahayn in borotiinada plasma. Waxaa ku hadla ku saabsan waxtarka. Tan iyo factor yar ku qabanaya, daawada waxaa ka fiican u nuugo. Dhigaalka waa kelyaha, beerka, ee unugyada muruqa, ee qanjidhada dhareerka ah. In jidhka, metformin isma badelin. Waxa uu markii dambe saxarrada kelyaha. Sidaa darteed, in ay dhacdo xadgudub ku ah shaqadooda lagu arkay raasamaal. Biological bar-nolosha waa 1.5-4.5 saacadood.
aayahooda
Daawo "Formetin" waxaa loo isticmaalaa daaweynta ee qaybaha qaar ka mid ah cudurada. Magac ahaan, iyadoo ay wada joogaan ee macaanka nooca II, kiisas cayilka leh u adag marka cunto uusan caawin in ay sii heerka sonkorta dhiigga caadiga ah, xataa isku dhafan oo sulfonylurea ah. Sidoo kale wax ku ool ah waa "Formetin" waayo, miisaanka oo yaraada.
Sida loo qaado?
Qiyaasta dhakhtarka loola jeedaa sooco, oo ku salaysan cadadka of glucose ee dhiiga. Maamulka Afka lagama maarmaan ah in ay gutaan cuntada ka dib, la cabo xaddiga badan ee dareeraha ah iyo tiriska machining kiniinka. Sida aynu hore u kor ku xusan, qiyaasta loo qoro ku xiran tahay content ee sonkorta ee dhiiga. Waxay ku bilaabmaa lacagta ugu yaraan - 0.5 g ama 0,85 g maalintii. Laba maalmood ka dib daawaynta bilaabin la daroogada this ayaa content joogta ah metformin ee dhiigga. Optionally, si tartiib ah u sii kordhaya qiyaasta ilaa qiimaha ugu badnaan. Waxay u dhigantaa 3 grams.
Tan iyo dadka waayeelka ah inta badan lagu arkay horumarka aysiidh jėrto, iyaga, waayo, heerka qiyaasta ugu badan ee maalin walba ah ee lacagta 1 g of daroogada waxaa sidoo kale hoos u xadgudub shiid, si looga hortago dareen xaasaasi ah, taas oo u muuqato in foomka of finan maqaarka, iyo dhacdooyin kale oo gurracan ee suurogalka ah, kaas oo lagu qeexay doonaa hoos.
sababo
Marka tan la eego, waxaa jira Gudigga badan. Drug "Formetin" tilmaamaha loo isticmaalo taasoo lagu muujiyay qoraalkan, waa u ay goobjoog ka ahaayeen:
- ketoacidosis Diabetic, precoma, kooma.
- shaqeynta kelyaha daran si daciif ah.
- failure Wadnaha iyo neefsashada.
- wajiga Ba'an ee Wadnaxanuun myocardial.
- Fuuqbaxa.
- Khamriga Chronic iyo xaaladaha kale ee laga yaabo in ay ka qayb qaataan muujinta horumarinta aysiidh jėrto.
- stroke Ba'an.
- Uurka iyo naas-nuujinta.
- Diidmo in srudstvu this.
- qaliin Major ama dhaawac, markii insulin waxaa loo doortay.
- cudurrada faafa daran.
- xanuunada Functional beerka.
- sumowga Xiisad khamriga.
- aysiidh melkesyrebakterier (oo ay ku jiraan taariikhda).
- cunto Hypocaloric (in ka yar 1000 Kcal. maalin Per).
- Adioizotopnyh ama waxbarasho radiographic, maamulka nooca iodide walax.
Waxaa sidoo kale aan lagu talinayaa in la isticmaalo daroogada "Formetin" qof ka badan lixdan sannadood, qabashada shaqada jidh ahaan culus. Tan iyo markii ay dhacdo in this, waxay leeyihiin halis kordhaysa oo ah horumarinta aysiidh jėrto.
dhibaato
dhacdo ee calaamadaha aan fiicneyn sida dhadhanka "macdan ah" afka, matag, yalaalugo, shuban, yaaqyaaqsi, rabitaan la'aan cunto u baahan joojiyo isticmaalka daaweynta iyo gudbinta deg deg ah ku takhasusay. Isticmaalka muddada dheer ee daroogada sababa qas ama joojin buuxda oo ku qaadashada of vitamin B 12, taas oo horseedaysa in ay raasamaal ee jirka ka mid ah dambe, taasoo keenta yaraanshaha vitamin. Marar dhif ah, dambe soo koraya - megaloblastic anemia 12-yar. Haddii si khaldan ay maamusho dose hypoglycemia suurto gal. Waxa kale oo aad la yeelan karaa xasaasiyad sida finan maqaarka. Sidaa darteed, daroogada dib u eegista "Formetin" kaas oo ay ku habboonaanta in isticmaalka kala duwan, waa in la magacaabay oo kaliya uu dhakhtarka xaadirka ah.
ganaaxyada
Muqaalka muhiimka ah lagu qeexay shuruudaha kaydinta walax aasaasiga ah "Formetina" ee jidhka iyo natiijo ah oo this.
Si looga hortago raasamaal aysiidh jėrto iyo ka hortagga metformin, waxaa lagama maarmaan ah in lala socdo tusayaasha ee shaqada kelyaha iyo baaritaan si loo ogaado waxa ku jira jėrto ee jirka ku jira ugu yaraan 2 jeer sanadkiiba. Sidoo kale, haddii aad leedahay xanuun muruqyada waa in la baadho.
Raad ku sheegay daroogada on awood u leh inay la wado farsamooyin iyo kaxeeyo
Xaaladdan oo kale, maadaama ay jiraan Gudigga qaarkood. Impact "awoodda Formetina 'in ay ku shaqayn mishiin iyo gaadiidka qaadataa meel keliya haddii lala isticmaalaa daawooyin saameeya geedi socodka shaqo u baahan in xawaaraha jawaabaha oo kordhay ka -fiirsashada. Waxaa muhiim ah in la ogaado.
Codsiga uurka iyo nuujinta
Diyaarinta "Formetin", tilmaamaha isticmaalka kaas oo lagu qeexay, taasina, waxay leedahay saamayn on caloosha ku category «B» by FDA. Inta lagu guda jiro uurka heli kartaa lacag this. Si kastaba ha ahaatee, ay la isticmaalo wuxuu noqon karaa oo keliya xaaladaha qaarkood. Oo kuwaasu - marka natiijada ka therapy this filayaa badnaan doonaa helitaanka halista ka iman karta in ilmaha caloosha ku. waxbarashada gaarka ah iyo kiis ku saabsan isticmaalka qalab sida daroogada ah "Formetin" la sameeyay muddada uurka. Waqtiga daaweynta waa in ay joojiyaan naasnuujinta. Si kastaba ha ahaatee, waxaad u baahan tahay inaad la tashato dhakhtar aqoon u leh.
isdhexgalka daroogada
Metformin kordhiyaa heerka sonkorta dhiigga. Tani gaar ahaan waa cad la soo dhaweynta isku mar ah daawooyinka aan steroid ahayn anti-bararka, taagayo sulfonylurea iyo clofibrate, inhibitors oxidase monoamine, acarbose, insulin, oxytetracycline, cyclophosphamide, inhibitors ee angiotensin diinta blockers enzyme iyo nooca.
Marka wada codsatay daawooyin hormoonada (piller, corticosteroids, sympathomimetics epinephrine, hormoonnada qanjirka thyroid, glucagons, thiazide iyo "loop" diuretics, taagayo phenothiazine, taagayo acid nicotinic) metformin laga yaabaa in habka Fariin hypoglycemic.
Iyada oo isku-dar ah qalab sida daroogada ah "Formetin" with "Tsimidinom" "nifedipine" khatarta sii kordhaysa ee aysiidh jėrto, metformin anada Digo jidhka ka. Noocan oo kale ah lagu arkay shaqo ee wax soo saarka khamri, in H. Vol. In ka kooban daawooyin ah.
wakiilada Cationic (quinidine, amiloride, digoxin, procainamide, morphine, quinine, vancomycin, ranitidine, triamterene) sameeyay tubules ah, tartamaya nidaamka gaadiidka iyo daaweyn muddo dheer kordhin kartaa heerka fiirsashada daroogada in 60%.
badinta
Iska badinta "Formetinom" arkay marka la qaadanayo 0,85 garaam maalin kasta oo ka cadhaysiinina aysiidh jėrto. Sidoo kale, content sare ah metformin sabab u ah kelyaha.
Calaamadaha ugu horeeya ee aysiidh jėrto waa itaaldarrada jidhka oo dhan, dibiro, heerkulka jirka oo hooseeya, xanuun caloosha iyo muruqyada, cadaadis dhiig oo hooseeya, bradyarrhythmia reflex. Xaaladaha qaarkood, waxaa jira daliilka soo noqnoqda ee cudurada neef-mareenka, dawakhaad, iyo, sida natiijo ah, waxaa jira horumarinta kooma.
At ugu yar ee calaamadaha ah qiyaasta xad dhaafka ah waa in joojiso isticmaalka daroogada iyo la tasho dhakhtar si loo xaqiijiyo cudurka aysiidh jėrto. Waayo, ka saarida oo ah walaxda firfircoon oo ka mid ah wakiilka iyo jėrto ka shaqeeyo ah kelyaha doonaa barbar daaweynta calaamadaha.
"Formetin": dhigooda
Waxaa jira wax badan oo ka mid ah ilaha dhaqaale ee noocan ah. Analogues "Formetina" taag daawooyinka ay ku jirto sida qayb weyn ee hydrochloride metformin in ay ka kooban. Mid ka mid ah tusaale ahaan waa daroogada ah ee soo saarayaasha Ruush, "Vero Metformin," "Gliformin", "metformin", "Metformin-Richter", iyo dibada - "Glucophage", "Glucophage" iyo "Glyukofazh Long" (France), "Lanzherin "(Slovakia)" Metfogamma "la qaadashada oo ah walaxda firfircoon ee 0,100, 0,500 iyo 0,850 g (Germany) kala duwan.
Xaaladaha iyo shuruudaha
Marka tan la eego, waxaa jira shuruudo gaar ah. Diyaarinta "Formetin" waa awood a, sidaa darteed waxaa la sii daayay oo keliya by qoro oo u baahan kaydinta heerkulka qolka, out of carruurtu gaari karin iyo meel iftiinka qoraxda. Shelf waxaa nolosha - 2 sano.
qiimaha
Qiimaha caadiga ah ee daroogada "Formetin" ayaa lagu wadaa ku xiran qiyaasta ka 59 rubles. 0.5 g of khariidad, 133 rubles. of 0,85 g iyo 232 rubles. in ka badan 1 sano
gunaanad
qorani oo dhan waxaa ka mid ah macluumaad badan oo faa'iido leh. Ka dib markii reading this article, qof walba inuu awoodo inuu helo jawaab su'aasha ah ee sida loo qaato 'Formetin "iyo waxa uu leeyahay sifooyin u noqon doonaa.
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