Caafimaadka, Diyaarinta
Daawada "Akineton": tilmaamaha loo isticmaalo, sharaxaad, dib u eegista
walaxda firfircoon "Akinetona" waa hydrochloride biperiden. Tablet caawinaysa 2 mg oo ah walaxda firfircoon. Intaas waxaa sii dheer, joogitaanka qaybaha dheeraad ah (galleyda, istaarijka baradho, laktosmonohydrat lactose, milmahayn magnesium, cellulose mikrokristallin, copovidone, calcium hydrogen dihydrate phosphate, Rusheyn kartaa, biyo daahir ah) qabanayaa daroogada "Akineton".
Tilmaamaha loogu isticmaalo, sawirka soo jeedisay in qaab kiniin oo ah daroogada uu leeyahay ficil ahaan midabka cad, qaab Valium. On hal dhinac oo kiniin ah waxaa jira halis of a beveled iskutallaabta qaab.
1 ml of xal ku jira lactate biperiden qadarkuu of 5 miligaraam. Qaybaha dheeraadka ah waa: duro biyo iyo sodium lactate.
saamaynta pharmacological
biperiden qayb Main - holinoblokator tallaabo dhexe.
Saamaynta ay ku lug leedahay diiqadoodo awood u leh inay hawl neuronal cholinergic in striatum ah, taas oo ah unugga dhismaha nidaamka extrapyramidal.
daroogada wuxuu keenaa saamayn ganglioblokiruyuschimi, darnaanta saamaynta m-anticholinergic maroojiska oo dhexdhexaad ah ee ubucda (maroojiska).
Isticmaalka daroogada ka caawisaa baabi'iyo gariirka addinka, kaas oo soo baxdo in isticmaalka daroogada cholinergic (tus, pilocarpine) iyo catalepsy iyo rigidity muruqa in bukaanlayda qaadato neuroleptics. Waxa uu awood u leeyahay si ay u abaari cadhoodaan.
Pharmacokinetics
"Akineton" xidhxidhan borotiinada plasma at 91-94%. ansixin Plasma noqon doona 11.6 ± 0.8 ml / min / kg miisaanka jidhka. Hal dose oo ah dejinta afka ayaa bioavailability ah oo ku saabsan 33 ± 5%.
Galaa caanaha naaska.
Biperiden buuxda metabolized ee jirka aadanaha. In kaadida, walax aan la go'aamiyo qaab oon doorsoomaynin. The metabolites waaweyn yihiin bicycloheptane iyo piperidine, kuwaas oo ah wax soo saarka ka saxarada iyo kaadida.
Elliminatsiya fuliyay laba weji, iyadoo nolol bar (1/2 T) ee 90-ka daqiiqo lagu jiro wajiga koowaad iyo 24 saacadood - wajiga labaad. In bukaanka dadka waayeelka ah, badhkiis nolosha kor u qaadi kara si xooga.
Tilmaamayaasha
"Akineton" loo isticmaalo xanuunada extrapyramidal laaluusheen by Maamulka daawooyinka qaarkood (neuroleptics, jirada dhimirka).
Sidoo kale, daroogada waxa lagu tilmaamayaa lagu ogaado cudurka Parkinson ee syndrome, parkinsonism (wakiilka maamula ee therapy isku dhafan oo saldhig a)
sababo
Ujeedada daroogada this aan la muujiyey marka aad xasaasiyad in ay qayb firfircoon ee daroogada "Akineton".
Tilmaamaha loogu isticmaalo wargelinaysaa in daroogada waa in laga fogaadaa sida wayneeyo prostate, gulukooma xagal-xidho, isbedel obstructive ee xiidmaha (stenosis pylorus, Bilowgii ileus curyaanka) in lagu ogaado xanuunka ee bukaanka ah.
Arrhythmia, qalalka, quudinta naaska, waayeelka, uurka waa arrimo kuwaas oo "Akineton" maamulay si taxadir leh u weyn.
waxyeellooyin
waxyeelo habdhiska dhimirka waxaa lagu muujiyey asthenia, daal, feejignaan xumo, daciifnimo, kabuubyo, dawakhaad, dareen walaac, walwal, dhantaalan xasuusta, wareer, dhalanteed, catalepsy, daroogada ku tiirsanaanta daroogada "Akineton".
Tilmaamaha loogu isticmaalo hadalka ku saabsan dhibaatooyin soo raaca oo qayb ka mid ah aragtida ah - mydriasis, qas hoyga.
nidaamka wadnaha-vascular waxa lagu gartaa dhaqsad heerka garaaca wadnahaaga ee (tachycardia); mararka qaarkood - deceleration (bradycardia); markaad codsanayso qaab cirbad diyaarinta - hoos u cadaadiska dhiigga (hypotension).
On qayb ka mid ah nidaamka dheefshiidka - afka oo qalala, calaamadaha dyspeptic, calool.
On qayb ka mid ah dheef - hoos u dhidid.
On qayb ka mid ah nidaamka kaadi - in bukaanka qaba wayneeyo (hypertrophy) ee qanjirka 'prostate' - dhib suurto gal kaadida.
cadaanyo: finan maqaarka, cuncun.
Hababka Isticmaalka
Waayo, muruqyada dhexdooda, xididka, iyo kiniin afka waa diyaarinta taam "Akineton".
Tilmaamaha loogu isticmaalo jeedisay in therapy "Akinetonom" guud ahaan wuxuu bilowdaa ka yar ka qaataan, qiyaasta more korodhka stepwise ku xiran tahay saameynta doonayo daweynta iyo waxyeellooyin.
Dadka waaweyn ee isticmaalka foomka afka ah ee diyaarinta bilaabin daawada at dose oo ah 1 mg 1-2 dhaweyn inta lagu jiro maalintii ama 2 mg qaybiyay laba qaadasho maalin kasta. Dheeraad ah, qiyaasta waa la kordhin karaa ilaa 8 mg laba ilaa afar qaadasho kala. Si kastaba ha ahaatee, qiyaasta waa in aan loo kordhiyo wax ka badan 2 mg maalintii. Ha ka badan qiyaasta ugu badan waxay ka dhigan tahay 6 galay Th-16 mg muddo shan maalmood ah. foomka daroogada la isku duro hal dose waa in aanay ka badan 2.5-5 mg. dose Tani yaabaa in lagu celiyo ka dib markii nus saac ah, laakiin tirada maamul maalin kasta waa in aan ka badnayn 4 jeer. Qiyaasta ugu badan ee medicament qaab isku duro waa 20 mg muddo shan maalmood ah. Marka qiyaas fiican laga gaadho, ka dibna kala guurka ah si ay u soo dhoweynta "faafiyo Akinetona."
Laakiin ha iloobin oo ku saabsan hab qofka bukaan kasta ee therapy biperidenom ballanta.
cudurada extrapyramidal timi sabab u qofku cuno daawooyinka qaarkood (jirada dhimirka ama neuroleptics) waxay u baahan tahay shaqo walax la siiyaa qiyaas hal of 2 mg oo afka ah ama parenterally. Maamulka celi dose ayaa sheegay in waxa laga yaabaa in saacad kasta bar. Si kastaba ha ahaatee, sida kor lagu soo xusay, tirada maamul waa in aan ka badnayn 4 jeer. Qiyaasta afka waa in la kala qaybiyaa hal ilaa saddex qiyaasood.
cudurka Parkinson waxay ku lug leedahay maamulida daawada afka at 6-8 mg in 2-4 qaadasho kala qaybsan for maalin, qiyaasta lagu si tartiib tartiib ah kor u kordhin karaa inay tahay 6-16 sano mg.
Carruurta ka yar sanad ujeedada soo jeedinaya suurtagalnimada ee daroogada ee foomka isku duro si tartiib tartiib ah, dhoos keli ah 1 mg ama 0.2 ml. Marka da 'ka hal sano ilaa lix sano maamula 2 mg ama 0.4 ml. Laga soo bilaabo 6 ilaa 10 sano - 3 mg ama 0.6 ml. dose Tani yaabaa in lagu celiyo ka dib markii nus saac ah la degdegga ah. In joogitaanka waxyeello ka soo gaartey maamulka daroogada waa in ay ahaataa isku duro joojiyey.
Inta lagu guda jiro foomka afka ah therapy daroogada ee da'da 3 ilaa 15 sano qaadashada qiyaasta 1-2 mg in 1-3 saacadood inta lagu jiro maalinta.
Kiniinnada Iskuma wada cabbi kartaan calool madhan, oo waa in aad cabto qadar dhexdhexaad ah oo biyo ah. At dhacdo of waxyeelo aan loo baahnayn ka habdhiska dheefshiidka waa in ay qaataan daawada isla markiiba cuntada ka dib, yaraynta darnaanta saameynta xun loola jeedaa "Akineton".
Tilmaamaha loogu isticmaalo waxay muujinaysaa in in ay dhacdo sumowga nicotine ee dadka waaweyn ee caadiga ah therapy adag ayaa sidoo kale maamula daroogada this, iyo qiyaasta waa 5-Th-TB-10 mg noocyada isku duro, laakiin kaliya in kiisaska halis nolosha bukaanka.
Marka khubad isku fosfooraska organic kacmaha biperiden waxaa lagu fuliyaa si gaar ah ku xiran tahay darnaanta lesions. Ka bilow qiyaas 5 mg in ay dhacdo maamulka xididka, maamulka noqnoqda sii ilaa calaamadaha baaba'aan sumowga.
badinta
Iska badinta teedu saamaynta anticholinergic fahmayaan sababa daawada "Akineton".
Tilmaamaha loogu isticmaalo, dhakhaatiirta dhab ah bixiso si ay xaqiiqada ah dareenka in daaweyn jiray posimptomnaya xaaladan (dayactirka wadnaha iyo nidaamka neef-mareenka, daweynta oksijiinta, iyo hagaajinta hyperthermia, go'an tuubada kaadida, haddii loo baahdo). U baahan hordhaca ah ee inhibitor cholinesterase ah (physostigmine horrayn) .
dhexgalka
"Akineton" halka isticmaalka m-holinoblokatorami, daroogada isagoo antihistamine ah iyo ficil antiepileptic wanaajisaa hadal doonana. Si kastaba ha ahaatee, codsi isku mar ah metoclopramide yaraynaysaa saamaynta ay ku daweyn. Waxaa incompatibility daroogada kama dambaysta ah la ethanol. Ballanta quinidine kordhay jeer halista calaamadaha Tardive. saamayn M-cholinergic waa wanaajiyey markaad codsanayso levodopa.
Kaydinta iyo sale
Si aad u iibsato daawada waxay u baahan tahay warqad si ay u bixiyaan farmashiistaha. Si aad u kaydiso "Akinetona" waxay u baahan yihiin in ay u hoggaansamaan heerkulka, t. Heerkulka E. daarmayaay'e waa in aanay ka badan 25 digrii (qiyaasta Celsius). Waxaan u baahanahay meel aysan carruurta xarunta "Akineton".
Buugga nooleeya shelf ee daroogada ah - shan sano.
ganaaxyada
Magacaabidda biperiden xilliga uurka iyo nuujinta (nuujinta) wuxuu u baahan yahay tilmaamo adag.
Biperiden heli kartaa ilmaha caanaha naaska, Daalin ku meel gaar ah ee naas-nuujinta si ay u sii wadis la'aanta ah ee daroogada "Akineton".
description Product tilmaamay, in go'aan ku saabsan magacaabidda biperiden xilliga uurka iyo nuujinta tixgeliyaan halista ka iman karta in ilmaha, ilmaha caloosha.
Waayeelka noqdo arrin halis ah oo lagu daweeyo daroogada this a. Sidaa darteed magacaabi "Akineton" kooxdan oo ah dadka si taxadir leh u weyn.
Maqnaanshaha Kickaha cadaymaha mid ka mid ah isticmaalka ammaanka ee carruurnimada, waa sababta aan codsan carruurta daroogada "Akineton".
Description of diyaarinta (diiwaanka) ku qeexan yihiin xaqiiqda ah in digniin loo baahan yahay marka la isticmaalayo daroogada this bukaanka qaba qalalka ama aamba.
Iyada oo la isticmaalo daba dheeraaday waxa dhici karta ku tiirsanaanta daroogada.
Halista bixitaanka syndrome ku lug leedahay joojinta tartiib ah therapy "Akinetonom".
isticmaalka cabitaanka khamriga ku jiro waa in laga fogaadaa inta lagu guda jiro therapy ah.
Daaweynta la daroogada this u baahan waayana ka wadista baabuurta iyo isboortiga hawlaha u baahan-fiirsashada sare iyo jawaab psychomotor degdeg ah, tan iyo markii ay xambaarsan tahay waxaa la khatarta ka iman karta sabab u halista ah ee wareer.
"Akineton". Tilmaamaha loogu isticmaalo. analogs
Micne ah ee diyaarinta yihiin walxaha soo socda: "Biperiden" "Mendileks" "hydrochloride biperiden".
"Akineton". Reviews
Daawada waa heer sare ah wax ku ool ah in daaweyn jiray gariir Parkinsonism ee addinka la joojiyo ka dib ah oo waqti gaaban. Ayaa sheegay in si fiican loo dulqaadan daroogada "Akineton".
Jawaab-celinta forums ah hadalka ku saabsan suurtagalnimada of muujinta qaar ka mid ah waxyeelo inta aad qaadanaysid daawada.
Price "Akinetona". halkaas oo ay u soo iibsadaan
Qiimaha xalka laga yaabaa in ku dhawaad 800 rubles.
Price dejinta afka "Akinetona" - 560-580 rubles.
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