Caafimaadka, Diyaarinta
"Artrozan": tilmaamaha loo isticmaalo
tilmaamaha "Artrozan" loo isticmaalo waxaa loola jeedaa qaybta bukaan eegida iyo pharmacological of oxicams. The walax ugu weyn ee firfircoon ee diyaarinta - meloxicam in uu yahay wax ku ool ah oo la xushay Cox-2 inhibitor. Cinwaan looga dhigay "Meloxicam" daroogada this ka diiwaan gashan diiwaanka of INN.
Foomka kiniin oo ah daawada la sameeyo galay kiniin ah oo miisaankeedu yahay 15 mg ama 7.5 buuxiyey galay finan Electricity dusha.
By daawada guryaha pharmacological "meloxicam", oo lagu soo jeeda walax enolievoy acid, hab ficil anti-bararka iyo xanuunka. Hannaanku wuxuu ku salaysan yahay awoodda daroogada si uu xakameeyo socodka ah ee synthesizing prostaglandins. Under saameynta ay falcelin daroogada dhacdaa, inta lagu guda jiro kaas oo eegista joogsada waxqabadka of Cox-2 ensaymes, taas oo qayb biosynthesis ugu weyn qaadan.
Iyadoo qaadashada daroogada, guide "Artrozan" sharxayaa ay tallaabo hab this. Haddii daawada la maamulo ee qaadasho sare, ka dibna inta lagu guda jiro muddo dheer ay la isticmaalo waxaa hoos u dhac in selectivity ee Cox-2. Daawada ka yar saamayn ku Cox-1, kaas oo ilaaliya mareenka caloosha iyo mindhicirka. Taasi waa ay sabab u tahay tallaabadan la xushay iyo ilaaliyo mareenka caloosha iyo mindhicirka ka erosive iyo lesions kolit.
saamaynta daroogada anti-bararka The "Artrozan" diiwaanka xidhiidhsan xakamaynta dhaqdhaqaaqa enzyme of Cox-2, kaas oo u dhaqmo in koorsada ee geedi socodka bararka.
Pharmacokinetics "Meloxicam" waxa lagu gartaa sida soo socota. Qaybinta "Artrozan" awoodaan in ay ka gudbaan caqabadaha ay jidhka-cadka, ay sabab u tahay xarunta la borotiinada plasma u sarraysaa sida 99%. Halabuurka The oo qiimo synovial fiirsashada dheecaan kiiskan waa 50%.
-Shiid: daroogada ayaa ku dhowaad si buuxda u metabolized in unugyada beerka, sidaas waxaa jira formation of dhowr taagayo pharmacologically dhexdhexaad ah.
Digo: The soo saarka "meloxicam" muujinaysaa ku saabsan saamiyada loo siman yahay inta badan in ay kaadida iyo saxarada qaab alaabta dheefshiidka. % Ka mid ah qaybaha kaliya 5 waa wax soo saarka ka soo xiidmaha.
The guryaha pharmacokinetic ah "Artrozan" Buuggan daroogada waxbarashada ayaa sidoo kale go'aaminaya waayo, xaalado gaar ah. Gaar ahaan, bukaanka dadka waayeelka ah marka la helo ansixin hoos daroogada, iyo in ay dhacdo astaamaha cagaarshowga iyo renal failure, daroogada waa saamayn aan qiimo lahayn on pharmacokinetics ah.
Diyaarinta "meloxicam" waa si fiican u nuugo ka soo mareenka caloosha iyo mindhicirka, bioavailability ee ay heer gaadho 89% oo aan la saameeyeen cunto qaadashada. Reception at qiyaasood dose soo saaray bixisaa fiirsashada saami ka mid ah daroogada ee jirka.
Qaybinta: Sida caadiga ah, qaab aan fiicnayn CSS dhici on saddexaadna wuxuu u soo maalinta shanaad ee daaweynta, halka isticmaalkeeda muddo dheer waxaa la siiyaa uruureen deggan dhigma soo koobin pharmacokinetic hore.
qiyaasta of daroogada "Artrozan 'tilmaamaha loo isticmaalo waxaa lagu go'aamiyaa sida soo socota.
Codso daroogada ee foomka marka la isku daro lagu talinayaa. mudada lagu taliyey:
- in marxaladda hore ee daaweynta, 2-3 maalmood, codsatay "Artrozan" -ukoly;
- saddex ama afar maalmood maamulka muruqyada dhexdooda ka dib waa u guuraan si ay u helaan daawo afka - qaab kiniin.
qiyaasta maamulka muruqyada dhexdooda, iyo maamulka afka la mid yihiin oo loo siman yahay heerka (7.5 ama 15 mg) hal mar maalin maalmaha. The dose iyo mudada codsiga go'aamiyo xooganaanta ee xanuunka iyo heerka darnaanta ee caabuq. Si loo go'aamiyo qiyaasta waa in si taxadir leh loo tixgeliyo khataraha ka iman kara dhibaatooyin ka mareenka caloosha iyo mindhicirka.
In joogitaanka kelyaha, qiyaasta maalin kasta ugu badan ee aan ka badnayn 7.5 mg.
Isdhexgalka daawooyin kale oo la mid adag waxaa laga yaabaa in ay dhacdo ee saamaynta erosive-qoon leh ee mareenka caloosha iyo mindhicirka. Ha qaadan daawada xilliga uurka iyo nuujinta.
Product "Meloxicam" waa in la ilaaliyo, meel gudcur ah, waayo wax ka badan laba sano.
Drug iibin by qoro oo keliya.
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