Caafimaadka, Diyaarinta
"Theophylline": tilmaamaha loo isticmaalo, analogs
Sidee baan u isticmaalaan daroogada "Theophylline"? Tilmaamaha loogu isticmaalo, analogs iyo sifooyinka of lacag la dambe hadli doonaa.
The Halabuurka iyo qaabka
Taasi waxaa ku jira daawada, "Aminophylline"? Tilmaamaha Isticmaalka dhigayaa in element firfircoon ee qalab kanuna waa magaca la mid ah walaxda - aminophylline.
Daawada waxaa suuq sidii xal loogu talagalay maamulka xididka, iyo sidoo kale qaab kiniin, labeen ama boomaato.
Tilmaamo pharmacological
Waa maxay daawaynta sida "Theophylline"? Tilmaamaha loogu isticmaalo (ampoules daroogada this laga iibsan karaa farmashiye kasta) ayaa sheegay in ay tahay vasodilating, maroojiska, durayo iyo daroogada bronchodilatory.
element firfircoon ee medicament waa cusbo ah ethylenediamine theophylline. Waxay saamayn bronchodilatory iyo bronchodilator ah, ay sabab u tahay saamaynta relaxant toos ah on fiiloyin vascular muruqa siman ee sambabada iyo marinada hawada. saamayn Tani waxaa sababa Iscelin ee la xushay ee hawsha phosphodiesterase, taasoo keentay in koror xerada intracellular.
sifooyinka daroogada
Qalab cajiib ah "Theophylline"? Tilmaamaha loogu isticmaalo sheegayaa in uu awoodo in uu yareeyo hyperreactivity ee neef-mareenka. hab ay ficilkan weli la aqoon, laakiin khubarada ayaa sheegaya in isticmaalka daroogada loo arkaa sababa in la kordhiyo tirada iyo hawlaha of T-suppressors ee dhiigga.
Kordhinta ansixin mucociliary, sii kordhaya foosha ee diaphragm ka, iyo sidoo kale madadaalo shaqada murqaha neefsashada intercostal, qalab shidaa xarunta neefsashada, caawiyo si loo hagaajiyo ay dareen, iyo wanaajisaa hawa alveolar, kaas oo ugu dambeyntii keenta in hoos u dhac ku badnaanta iyo adkaanta dhacdooyin xibin gal.
Sida saamayn kale ee daroogada ah, "Aminophylline"? Tilmaamaha loogu isticmaalo (cadar iyo xal leedahay saameyn la mid ah ku shaqeeyo) ayaa sheegay in hoos tixgelin ka dhigan tahay gacanta ku shaqo neefsashada, oon ku wanaajiyo qaabka robab O2 dhiigga iyo hoos u fiirsashada of carbon dioxide. Intaas waxaa sii dheer, daroogada firfircoon waa inay awoodaan inay kicin hawo ah hypokalemia.
Waa in la sidoo kale xusay in tilmaamaha "Theophylline" loo isticmaalo kaas oo hoos ku qeexan, qalbiga ku shidaa, waxay kordhisaa inta jeer iyo xoog of wadnaha ah, waxay kordhisaa baahida loo qabo in muruqyada wadnaha ee O 2 iyo si weyn u kordhiyaa socodka dhiiga ee wadnaha.
Isticmaalka dejinta this ka caawisaa si loo yareeyo midab cerebral vascular, kelyaha iyo maqaarka. Khubarada ayaa sheegaya in wakiilka loo arkaa tallaabo uu leeyahay venorasshiryayuschim durayo iyo durugsan hoos iska caabin vascular pulmonary, hoos u cadaadiska dhiigga ee wareegga pulmonary iyo dareen u socodka dhiigga kelyaha. Sidoo kale, dejinta this kor u mareenka biliary iyo caanuhu Amda dhiig xinjirowga sameeya iyo sii daayo ee dhexdhexaadiyayaal ka ah reactions diidmo, xasilinta derbigii unugyada waaweyn ee, dejisa microcirculation ah, yareeyo halista ah ee formation thrombus iyo hagaajinaysaa xasiloonida ee erythrocytes.
In qiyaasood oo waaweyn daroogada loo arkaa muujinaysaa guryaha epileptogenic.
kinetics
Waa maxay-beegyada uu caan ku ah hab "Theophylline" ogeed? Tilmaamaha loogu isticmaalo (slimming diyaarinta this waxaa loo isticmaalaa ilaa xad inta badan) dhigayaa in dib u shaqeeyo element aadanaha firfircoon ee daroogada la metabolized la sii daayo xiga ee theophylline furan, taas oo markii danbe xidhana borotiinka plasma in 40%.
Waxaa loo tixgeliyaa ka dhigan tahay awoodaan in ay dhex gasho iyada oo ka celiyaha mandheerta, iyo sidoo kale wax soo saarka caanaha hooyada.
theophylline Isbadal kordhiyay beerka by P450 cytochrome eulayska.
Foomka hore ee daawada waa wax soo saarka ee lacagta ah ee 10% in kaadida. Markii ugu bar-nolosha ee qalab this in aan sigaarka, iyo sidoo kale bukaanka ka cabanaya neefta bronki, waa 12 saacadood, in carruurta - 1-5 saacadood ee dhasha ah - ilaa 2 maalmood, iyo in dadka sigaarka cabba - 4 saacadood.
Marka ay maamusho?
Tilmaamayaasha for isticmaalka daroogada waxay ku xiran tahay qaabka ay sii daayo.
Maamulka Parenteral waxaa lagu talinayaa in:
- xanuunada ischaemic ah wareegga cerebral,
- asthmaticus status ,
- bidix ventricular failure, kaas oo ahaa mid adag oo ay cidhiidhi ku neefsashada, iyo bronchospasm;
- xibin gal dhalaanka;
- chronic oo ba'an wadnaha;
- bararka asal ahaan kelyaha.
Mararka qaarkood, iyadoo la isticmaalayo afka "Theophylline" (kiniin)? Tilmaamaha loogu isticmaalo warar sheegaya in qalab ay u qabata sidoo qalbiga ka pulmonary, syndrome broncho-obstructive of etiology kala duwan (tus, emphysema, neefta, COPD, boronkiitada obstructive), xibin gal, hurdo, cadaadis sii kordhaya ee wareegga pulmonary, wadnaha oo shaqadiisa gaba nooca daro ba'an .
sababo
Marka waa in aad isticmaalin daawada "Theophylline"? Tilmaamaha loogu isticmaalo warbixino in waa u in:
- barar aad u daran halbowlaha ama hypotension, tachyarrhythmia, boogaha of mareenka dheefshiidka, oo ay ku jiraan sii daridda ah;
- gastritis giperatsidnom, function kelyaha ama cagaarshowga daran, stroke dhiigbaxa, qalalka, hemorrhage in ileyska;
- isticmaalka isku mar ah ephedrine in carruurta da'doodu ka yar tahay 3 sano, kordhay dareen in aminophylline ama theophylline.
Drug "Theophylline": tilmaamaha loo isticmaalo
Cellulite (feedback bukaanka la hoos looga hadli doonaa) waa hab lagu caawiyo wanaagsan, laakiin tani ma aha ujeedada ugu weyn ee daroogada loo arkaa.
Sidee baan u isticmaali? mudada qiyaasta shakhsiga medicament. Daaweyntu waxay ku horumartay by dhakhtar khibrad leh ku xiran tahay sawir caafimaad, da'da bukaanka, iyo joogitaanka caddayn ku tiirsanaanta nikotiinka.
diyaarinta A qaab xal loo intramuscularly ama faleebo duri karo, iyo sidoo kale cadar - codsatay in nerazdrazhennuyu maqaarka qalalan.
Sida loo isticmaalo miisaanka oo yaraada?
Ma suurogalbaa in la isticmaalo daroogada miisaan lumis "Theophylline"? Tilmaamaha loogu isticmaalo (ee cellulite waa qalab inta badan loo isticmaalaa foomka ah oo cadar ku) ku jira saaraysa warbixin lahayn. Si kastaba ha ahaatee, khubarada ku doodaya in walaxda firfircoon ee daroogada this runtii waxay ka caawisaa si loo yareeyo miisaanka jidhka, laakiin sidoo kale qayb ahaan in laga takhaluso "diirka liin". Sidee tani u dhici? Xaqiiqada ah in aminophylline kobcin kara wareegga dhiigga ee nudaha ku, iyo sidoo kale in la hagaajiyo shaqada dheecaan ay. walax noocan oo kale ah oo laga helay dad badan oo kareemada for cellulite (tusaale ahaan, "Turboslim», Draine Minceur, Reflexe Minceur, Phyto-Complexe, Qaab-up , iwm).
Schematics ee codsiga of cadar la aminophylline ku xiran tahay oo sideeda oo buuxa iyo soo saaraha.
waxyeellooyin
Maxaa reaction ay dabiicadda ka soo bixi kara ka isticmaalka lacagta? Sida laga soo xigtay tilmaamaha, waxay keeni kartaa:
- hurdo xumo, walwal, dawakhaad, gariir iyo gariir,
- reflux gastroesophageal, matag, shuban, lallabo, laab, anorexia, iyo sii daridda cudurka boog ulcer,
- garaaca wadnaha, wadnaha xanuun, xaalad xumeyd ee kog, hoos u cadaadiska, angina been ah iyo tachycardia;
- hematuria, albuminuria;
- cuncun, xummad, iyo finan;
- hypoglycemia,
- barrar, xanuun iyo induration goobta la duray;
- tachypnea, albuminuria, xanuun laabta ah, hematuria, dareenka gubashada ah, hypoglycemia, dhidid iyo kaadida maalin walba kordhay.
Dhexgalka iyo badinta
Ilaa iyo hadda, Xaaladaha ayaa la soo sheegay hab farriimaha xogta badinta. Haddii xaaladda ay taasi dhacdo, waa in aad joojiso qaadashada daawada iyo daaweynta bilaabi astaamaha.
In isku midka ah qaadashada daroogada la sympathomimetics hawshooda u ah labada dhinac ee ay tallaabo pharmacological. Sida beta-blockers, iyo khayraadka lithium, falalka ku habboon yihiin labada wiiqay.
The saamayn "Aminophylline" daweynta sicad dhimay markii ay isku mar loo isticmaalaa la "pentobarbital", "rifamycins", "Isoniazid", "carbamazepine", "sulfinpyrazone," "phenytoin" (oo ay ku jiraan dadka sigaarka cabba).
Action tixgeliyo daroogada lagu kordhin karaa markii co-maamula la quinolones, "lincomycin" macrolides "cimetidine", "Allopurinol" isoprenaline, beta-blockers, fluvoxamine, piller, "Disulfiram", "Viloksazinom", iyo sidoo kale inta lagu guda jiro tallaalka hargabka .
Chelators iyo antidiarrheals yareeyo adsorption "Aminophylline."
Analogs iyo dib u eegista macaamiisha
Haddii ay jiraan analogs ah "Theophylline" daroogada? Khubarada jawaabi su'aashan jirini. daawo viewed bedeli kartaa "Aminophylline-esque", "Eufillin-Darnitsa", kiniin iyo irbado "aminophylline".
Maxay yihiin dad leh oo ku saabsan ayaa sheegay in ka dhigan tahay macaamiisha? Reviews of diyaarinta this waxaa jira waxyaabo badan ilaa xad ah. bukaanka intooda badan la sheegay in la isku duro "Aminophylline" waa qalab la xaqiijiyay. Its iyo hufnaanta ma keenaan wax shaki ah, oo ay ku jiraan weeraro xiiqda.
Sida for comments ku saabsan "Theophylline" cream, iyagu waa lagu muransan yahay. macaamiisha qaarkood waxay sheegeen in daawaynta tani waa natiijo la'aan. Si kastaba ha ahaatee, waxaa jira qaar ka mid ah bukaanka la wadaagi natiijada cajiib ah ka dib markii codsanaya cadar ee cellulite.
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