Caafimaadka, Diyaarinta
Drug "papaverine". Tilmaamaha kaa caawin doontaa in aad codsaneyso
Waxaa ka mid ah daawooyinka badan oo ku kalsoon in bukaanka sanado badan, waxaa jira daroogada sida "papaverine" sida. Guide qeexayaa si faahfaahsan oo dhan caddayn iyo heerka codsiga of dhimirka ah. In dabiiciga ah, walax tani waxaa ku jira xashiishad. Sanadihii la soo dhaafay, waxaa inta badan synthetically soo saaray. walax Tani - budada crystalline, wax yar L. ee khamriga, L. biyo si tartiib ah. Budada leedahay dhadhan yar qadhaadh. Xalka aqueous waxaa la hoos geliyey nadiifiye ah walax 0.5 saacadood at heerkul ah 100 ° C.
Drug "papaverine" waxa loola jeedaa miotropnym maroojiska. Waxay yaraynaysaa hawl contractile iyo yaraynaysaa midab ah ee muruqyada siman, waxay leedahay saamayn maroojiska iyo vasodilating. diyaarinta waxaa loo isticmaalaa sida calool maroojiska markii adkaashada murqaha siman a (waayo, cholecystitis, pilorospazme, ulcerös caydi, dubaaxin of mareenka kaadida), dhuumaha ugu sarreeya, bronki, weelasha maskaxda. Ilaa dhawaan daaweyso inta badan loo isticmaalaa si looga hortago istaroog. Qaadashada daawada edbinta "papaverine" oo ay ku jiraan macluumaad ku saabsan hantida wanaagsan, waa in la xusuustaa in qaabab sare, waxaa loogu talla tabinta intracardiac, yaraynaysaa excitability ee muruqa wadnaha. Daawada hoos u cadaadiska dhiigga.
Inkasta oo inta badan dhakhaatiirtu u qoraan daawada bukaan "papaverine", war aamusan oo ku saabsan xaqiiqada ah in farsamo ee ay tallaabo on jidhka bini'aadamka in dhamaadka weli unstudied. walax Tani - inhibitor phosphodiesterase a - Insaymkaas ah oo keena raasamaal intracellular xerada. Its raasamaal keenaysaa in hoos u dhac in muruqa iyo nasashada ee dalalka ay caydi.
Inta badan isku dhafan oo promedolom qoray macnaheedu yahay "papaverine" barashada kaas oo u ogolaanaya in aad u isticmaali isku dhafan oo daroogo kale bararka iyo xanuunka. therapy Tani waa in la baabi'iyo weeraro angina. Sidoo kale, waxaa inta badan qoray isku dhafan oo ah platifillin hab, phenobarbital iyo waxyaabaha kale.
Diyaarinta kiniin sii daayo "Papaverine" (0.04 g) ee baakado 10 kumbiyuutarada., In ampoules 1 iyo 2% xal of 2 ml, gelin dabada futada in 0.2 g walax firfircoon ee ku kiniin, si fudud cabaar dhex gistogematicalkie caqabadaha, si degdeg ah nuugo ka soo mareenka caloosha iyo mindhicirka. Daawada waxaa saxarrada kelyaha. Qeybtii - ka saac ilaa 2 saacadood. Ilaa 60% ka mid ah xal ah walaxda la sii daayay foomka xeryahooda kala duwan (glucuronic acid, phenolic).
Oo macnaheedu yahay "papaverine" edbinta oo si cad u muuqday, waxa qaadasho in ay qaataan daawada dadka bukaanka ah ee da'doodu kala duwan tahay, waxay u baahan tahay u hogaansanaanta adag in caadooyinka kuwan. qiyaasta xad-dhaaf ah inta badan keenta in cawaaqib xun. Dadka waaweyn ee maalin kasta waxaa caadi ahaan kuu qori 3-4 hal daawo dose 1 kiniin ah (0.04 g). U qoraan dadka kiniiniga ah ee carruurta, ku xiran tahay tirada sannadaha 3-4 dose hal qaadashada sida:
- 0.5-2 sano: 0.25-0.5 tab,.
- 3-4:. Table 0.5-1;
- 5-6: 1 tab,.
- 7-9:. Shaxda 1.5;
- 10-14: 1.5-2 tab.
Intramuscularly iyo subcutant duraa xal at 1-2 ml (1, 2%). Si taxaddar leh oo si tartiib tartiib ah ay maamusho xididka 2% xalka (2.1 ml), sida daroogada waxay keeni kartaa dhacdo ee block atrioventricular, aamba ventricular iyo extrasystoles ventricular. In foomka of saboostada la isticmaalayo hab ka mid ah 0,003-0,03 g dose hal (dose ku xiran da'da). Shumac loo isticmaalaa ka dib markii enema ama saxarada.
Qaadashada daawooyinka ahaan uu la darina diidmo, hypotension, xad gudub ku ah tabinta atrioventricular. Ha qaadan daawo aan la tashan dhakhtarkaaga. Waxtarka ama ay ammaanka xilliga uurka iyo nuujinta aan la aasaasay. Sidaa darteed, daroogada "papaverine" ah, oo tilmaan u ah oo codsiga ah ee xilligan ma waa u nolol, waxaa wanaagsan in aadan isticmaalin waa. Inta lagu guda jiro daawaynta mamnuucay qaadashada khamriga.
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