Caafimaadka, Diyaarinta
"Dipyridamole": tilmaamaha loo isticmaalo. "Dipyridamole": dib u eegista iyo analogues
Waa maxay daawada "Dipyridamole"? Tilmaamaha, qiimaha, qaababka, iyo tilmaamo ah lacagta lagu hoos lagu soo bandhigay doonaa. Waxa kale oo aanu kuu sheegi in ay macquul tahay in ay helaan ayaa sheegay in daawada inta ay uurka leedahay, haddii uu wax analogues, waxyeelo iyo sababo.
Curiska, xirxirida iyo qaabka
Oo muujinaysa in diyaarinta buugan edbinta? "Dipyridamole" - daroogada a in uu leeyahay nooc ka mid ah loo sii daayo. Kaalaya aan ka fiirsan in faahfaahin dheeraad ah:
- Dragee 0.075 iyo 0.025, walaxda firfircoon ee foomkan waa dipyridamole. Daawada waxaa lagu gadaa baakadaha caaga ah ee 100 oo gogo '.
- "Dipyridamole" - loox oo 0,075, 0,005 iyo 0,025 g dahaarka leh, waxay sidoo kale ka kooban walaxda firfircoon sida dipyridamole. Iyadoo la tixgelinayo waxyaalaha kaabayaal ah, tan dambe ayaa waxaa ka mid ah ku milmahayn calcium, laktosmonohydrat lactose iyo istaarijka. Daawada lagu iibiyo khariidad-120 ama 40 xabbadood, oo waxaa la geeyaa raso baakado.
- Xalka la isku duro. Foomkan waxaa ka mid ah walax la mid firfircoon. 0.5% xal lagu iibiyo fijaan of 2 ml.
pharmacodynamics
Waa maxay guryaha loo arkaa daawo? Maxay ku lifaaqan tilmaamaha loo isticmaalo? "Dipyridamole" - daroogada a in uu leeyahay saamayn vasodilating ah. tallaabo noocan oo kale ah waxa ay leedahay inta badan ee weelashii wadnaha.
qiyaasta aqbalay of medicament hakiyo Amda ee platelets siyaadiyaa heerka socodka dhiigga, hagaajinaysaa iyo Eebay tallaabo angioprotective. Waxaa intaa dheer, ay tahay maado kor wareegga rahaamad in weelashii wadnaha.
Waxaan ma dhihi karo in daawada normalizes dheecaanka arooriyaha. Sidaa darteed, ay qaadashada joogtada ah oo si weyn u yaraynaysaa khatarta thrombosis, gaar ahaan muddada postoperative.
Mabda 'hawlgalka
Waa maxay daawada kale wuxuu leeyahay sifooyin "Dipyridamole"? dalalka Buugga in ay ka dhigan tahay sidoo kale hoos u midab, oo weelasha cerebral. Marka tan la eego, waxaa ilaa xad si firfircoon loo isticmaalo weerar ischaemic. Waxaa intaa dheer, waxaa loo arkaa daroogada hagaajinaysaa wareegga sicad mandheerta. Habkaani wuxuu kuu ogolaanayaa inaad si looga hortago hypoxia uurjiifka.
Waa maxay hab ay of tallaabo daroogada? Waa maxay macluumaadka ku jira tilmaamaha loo isticmaalo? "Dipyridamole" kordhiyaa dhaqdhaqaaqa ee adenosine iyo yaraynaysaa unugyada gacanta ay. Ayaa sheegay in walax saamayn ku muruqyada vascular by xanibeen sii daayo norepinephrine, taas oo, dhab ahaantii, ka dhigi ay foosha, sii kordhaya cadaadiska dhiigga iyo iska caabin vascular systemic.
Sidoo kale waa in la ogaadaa in ay sabab u tahay ka xanibeen phosphodiesterase hoos u sii daayo xulkii activators ee platelets. Habkaani iyaga ka hortagtaa ka dusin. Hoos u dhaca adhesiveness dhiig xinjirowga ka hortagtaa xinjirowga dhiigga ee weelasha.
Drug "Dipyridamole", qiimaha kaas oo hoos ku qoran, sida wakiilada antiplatelet waxaa badanaa loo isticmaalaa isku dhafan oo acetylsalicylic acid.
Pharmacokinetics
Nuugo tixgeliyo hab si deg deg ah halkii. Its fiirsashada ugu badnaan la gaadho ku saabsan 60 daqiiqo ka dib markii maamulka.
raasamaal oo ah walaxda firfircoon waa la fuliyay in myocardiocytes. Drug Oo Qaliin-shiid beerka. In case of xadgudub jirka ah ee shaqada raasamaal ay suurtagal tahay.
Tilmaamayaasha
Medicament "Dipyridamole" qoray in cudurada soo socda:
- kaafi wadnaha dabiiciga ah ee joogtada ah,
- ka hortagga qabsamin of shunts iyo stents;
- angina,
- Wadnaxanuun myocardial (ma aha oo kaliya in wajiga ba'an);
- thrombosis arooriyaha iyo halbowlaha;
- stroke ischaemic;
- ka hortagga thromboembolism, gaar ahaan ka dib markii qaliin on wadnaha;
- kaafi mandheerta;
- encephalopathy wareegga dhiigga,
- atherosclerosis lugaha,
- xanuunada microcirculatory asal kasta;
- glomerulonephritis;
- Indvandrerrådgivningen in sepsis in ilmaha iyo toxicosis.
sababo
Sida laga soo xigtay tilmaamaha of lacag aan la isticmaali karaa haddii leexashooyinkaasi soo socda:
- hypotension ;
- angina deganayn,
- Wadnaxanuun myocardial ba'an;
- diidmo,
- garaaca oo daran;
- wadnaha decompensated;
- beerka,
- diathesis hemorrhagic,
- caloosha boogaha, gaar ahaan u janjeera in ay dhiig-bax.
Sidoo kale waa inaad ayaa sheegaya in daroogada taas waxaa loo qoray si taxadir leh in ay carruurta ka yar 12 sano jir iyo nuujinta. Intaas waxaa sii dheer, waa wax aan macquul aheyn in la codsado wakiilka intravenously inta lagu guda jiro burburkii.
Tilmaamaha loogu isticmaalo
"Dipyridamole" - daroogada anti-thrombotic ay tahay in la maamulo kaliya uu dhakhtarka xaadirka ah.
Guud ahaan, kiniin iyo kiniiniga afka laga qaato 60 daqiiqo cuntada ka hor, galaas oo biyo ah. In si loo yareeyo saamaynta ay diiqayo on xabka gastric daroogada la hoos dhiqi karaa caano diirran.
Qiyaasta iyo habka isticmaalka daroogada waa in la rakibo oo keliya by dhakhtar ku xiran da'da qofka bukaanka ah, akhriska iyo gobolka ee caafimaadka.
Waayo, ka hortagga thrombosis maamulo 75 mg ah medicament 6 jeer maalintii (dose maalin walba ugu badnaan - 300-450 mg).
Marka kaafi wadnaha iyadoo la isticmaalayo 25-50 mg oo daroogada ah saddex jeer maalintii. Qiyaasta ugu badan ee gobolka this - oo ku saabsan 150-200 mg.
Si looga hortago xinjirowga of jab stent iyo bukaanka la siiyo 50 mg daroogada (afar jeer maalintii) si wadajir ah ula acetylsalicylic acid. medicament waxaa loo isticmaalaa ka hor qaliinka, iyo sidoo kale inta lagu jiro toddobaadka ka dib.
Marka cudurada vascular occlusive ah addimada hoose waxaa lagu talinayaa in ay qaataan 75 mg ah ee daawada saddex jeer maalintii.
qiyaasta maalin walba ah ee daroogada si uu caruurta ku xiran tahay miisaankooda (5-10 mg halkii kg).
Sida laga soo xigtay tilmaamaha, inta lagu guda jiro daawaynta lagama maarmaan ah in la xaddido isticmaalka shaaha iyo kafeega, sida ay wiiqi karaan saamaynta daawada.
badinta
Marka la isticmaalayo qaadasho sare ee daroogada calaamadaha soo socda ee bukaan-socodka ah ayaa dhici kara: dhiig-karka, dawakhaad, garaaca wadnaha oo kordhay hoose iyo dhiig. Xaaladdan oo kale, loo joojiyo daawada iyo la tasho dhakhtar.
dhibaato
Sida laga soo xigtay jawaabaha dadka bukaanka ah, in xaaladaha qaarkood, soo dhaweynta ah ee lacagaha u keeni kartaa dhibaatooyinka soo socda:
- cadaanyo;
- wadno,
- hoos u cadaadiska dhiigga (gaar ahaan marka intravenously maamula);
- Torombositobiiniya;
- madax xanuun,
- xanuunada dyspeptic;
- qaylada madaxa;
- barrar wajiga,
- tachycardia;
- dhiig kordhay ama dhiig.
isdhexgalka daroogada
saamayn Antiplatelet daroogada waxaa lagu wanaajiyey maamulka isku mar la acetylsalicylic acid, tetracycline, penicillin, cephalosporin, xinjirowga lidka dadban iyo nicotinic acid.
Sidoo kale waa in la ogaadaa in aan toos ahayn xinjirowga lidka ku ah, thrombolytics iyo heparin kordhin kartaa suurtagalnimada dhibaatooyinka dhiig.
Waxaan ma dhihi karo in caffeine iyo xanthine daroogada yareeyo vasodilating iyo saamaynta anti-thrombotic lacagta, iyo laabjeexa yareeyo ay nuugista iyo in la yareeyo fiirsashada ee dhiigga.
Iyadoo la tixgelinayo diyaarinta tilmaamay, u kordhiyaa saamaynta maandooriyayaasha antihypertensive.
Ma isticmaali karaa daawada "Dipyridamole" inta aad uurka leedahay?
Khubarada ayaa sheegaya in inta aad qaadanaysid hoos tixgelin lacag haweenka uurka leh kulma dhibaatooyinka. On lid ku ah, "Dipyridamole" daroogada inta ay uurka leedahay waxaa inta badan qoray marka ay jirto halis ah dhicin ilmaha ahaan ama mandheerta.
Qiimaha iyo analogues
Daawada waxaa lagu beddeli karaa "Dipyridamole"? Analogs lacagaha hoos ku qoran. Kuwaas waxaa ka mid ah daroogada ee soo socda: "Parsedil", "Kurantil", "Padikor", "Antistenokardin", "Trankokord", "angina", "persantin", "Dipyridamole-Verein". Dhamaan daawooyinka waxay leeyihiin qayb ka mid ah oo firfircoon. Si kastaba ha ahaatee, waxaa laga yaabaa in ay qabaan waxyeelo kala duwan iyo sababo. In xiriir this, waxaa lagu talinayaa in la isticmaalo lacagta, kuwaas oo kaliya ka dib markii uu la tashado dhakhtarkaaga.
Waa imisa daroogada ah "Dipyridamole"? Its qiimaha u dhaxeysa 380-420 rubles (ku xiran cadadka iyo nooca daroogada loo sii daayo).
Reviews
Inta badan, aad warcelin oo ku saabsan qalab this hadhay kuwa bukaan kii laga soo qoray ee ka hortagga iyo daweynta dhicis gabowga mandheerta, iyo sidoo kale kaafi mandheerta.
Waa in la ogaadaa in dumarka uurka leh ku xanuunsado daroogada noocan oo kale ah waa fiican. Kaliya dhawr jinsi cadaalad ah isagoo dhibaato qaab hoos u dhac ku yimaadda cadaadiska dhiigga iyo wareer.
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