CaafimaadkaDiyaarinta

"Paroxetine": tilmaamaha loo isticmaalo, dib u eegista. analogues daroogada

Maxaa loola jeedaa daawada "Paroxetine"? Tilmaamaha isticmaalka daroogada loo soo bandhigi doonaa in this article. Sidoo kale soo baxay waxaa ka mid ah inaad ka warqabto kasta contra-tilmaamo iyo waxaa laga heli karaa daawo this, haddii uu lahaa waxyeellooyin, waxa foomka waa la heli karo iyo sida daroogada macaamila daroogooyinka kale.

Curiska, baakadaha iyo foomka of sii daayo daroogada

Drug "Paroxetine" tagaa on sale qaab kiniin, film-dahaarka leh. Waxay yihiin qaab wareeg ah oo lenticular, midabka cad, iyo khatarta ah ee dusha si adag.

walaxda firfircoon waxaa loo arkaa noo by loola jeedaa hemihydrat hydrochloride paroxetine. Sidoo kale, daroogada ee ay ka kooban leedahay qaybo taageero ah qaab ah Kolloidol dioxide Silicon, cellulose mikrokristallin, crospovidone, calcium phosphate hydrogen, copovidone, Rusheyn kartaa oo ku milmahayn magnesium.

Kiniiniga "Paroxetine" waxaa lagu gadaa baakad fin of 10 xabbadood oo waxaa la geeyaa kartoon ah.

tallaabada pharmacological daroogada

Waa maxay daawada "Paroxetine", taas oo analogues la sii magacaabi doonaa wax yar? Waa niyad jabka ah. Waa inhibitor ah ee neurons maskaxda reuptake (xulashada) serotonin. Tani waa waxa go'aaminaya ay saamaynta anti-niyad iyo oggolyahay ee daaweynta ee fawdo argagax iyo xanuunnada waswaaska.

Viewed xiriir medicament uu leeyahay xidhiidh ah oo aad u yar yahay α2-, α1- iyo β-adrenoreceptors iyo sidoo kale m-holinoretseptorami, dopamine, 5HT1-sida, 5HT2-sida iyo histamine H1-receptors.

Ma hawlaha psychomotor xadgudba daroogada "Paroxetine"? Reviews dhakhtarrada ayaa sheegaya in daawada saameyn ah kuma laha gunaanadeen aadanaha xun. Waxaa intaa dheer, waxa aanu potentiate saamaynta dejiye ee ethanol on hawlaha psychomotor.

La sheegay in cilmi-aqoonsaday niyad jabka ah guryaha kaakicin daciif ah sida kaliya haddii ay waxaa lagu qaataa qaadashada ka badan kuwa looga baahan yahay Iscelin of reuptake serotonin. Waxaan ma dhihi karo in daroogada this ma keeno isbaddal weyn ee heerarka cadaadiska dhiigga, EEG iyo garaaca wadnaha.

The pharmacokinetics qalab caafimaad

daroogada "Paroxetine" sida nuugo? Tilmaamaha loogu isticmaalo, dhakhaatiirta dhabta ah ayaa sheegaya in ka dib markii maamulka afka ah walaxda firfircoon nuugo ka soo mareenka dheefshiidka iyo waxaa metabolized dhex beerka.

fiirsashada taagan ee medicament dhiigga ku gaarayaa 1-1.7 todobaad ka dib bilow daaweynta daroogada. Walaxda firfircoon ee daroogada la ballaadhan loogu qaybiyey unugyo. Xaaladdan oo kale, waa boqolkiiba hal oo kaliya waxaa laga helaa plasma ah. Isgaarsiinta la borotiinada amarka of 95%.

Niyad jabka metabolized beerka. Sidaas darteed, metabolites firfircoonayn loo sameeyay. Waxay si dhakhso ah reebay jidhka ka, oo ay leeyihiin hawl yar pharmacological oo ay leeyihiin saameyn ah kuma laha waxyeelada daweynta of daroogada.

daroogada "Paroxetine" sida soo bandhigay? Fiiro gaar ah, farmashiistayaasha ratings sheegayaan in ku saabsan 64% oo ah walaxda firfircoon waa la soo wada saaro kaadida, halka 36% - in xiidmaha (in bile).

The pharmacokinetics daroogada xaaladaha caafimaad oo gaar ah

fiirsashada oo ah walaxda firfircoon ee plasma kordho dhiig xadgudub ku ah ee kelyaha iyo beerka, iyo sidoo kale dadka da'da ah.

Tilmaamayaasha ay u isticmaalaan qalab caafimaad

Xaaladaha qaarkood, bukaanka waxaa qoray niyad jabka "Paroxetine"? arjiga ku of guide qalab ku jira liiska soo socda ee akhrinta:

  • nooc kasta oo niyad-jabka, oo ay ku jiraan qoomiyadda daran, Waxyeelo, oo waxaa la socda walaaca,
  • argagixin xanuunada, oo ay ku jirto kooxda iscaawi;
  • disorder waswaaska (OCD ama soo gaabiyo);
  • ciladda wallaaca guud;
  • ciladda wallaaca bulshada, ama wax-u-cuqdadeedka bulshada.

Sababo in isticmaalka qalab caafimaad

Xaaladaha qaarkood, haddii ay dhacdo lahayn ma loo isticmaali karaa in bukaanka niyad jabka "Paroxetine"? arjiga ku of guide qalab ka mid ah liiska soo socda ee sababo:

  • qalalka deganayn,
  • isticmaalka waafaqsan of inhibitors oxidase monoamine, iyo sidoo kale muddo labo isbuuc ah ka dib markii ay ka bixitaanka,
  • da'da carruurta;
  • xilliga uurka,
  • Diidmo in qaybaha daroogada,
  • inta lagu jiro naas-nuujinta.

Isticmaal si taxadar leh u daran

In waxa Xaaladaha waa in la gacanta ku qaadashada ee lidka diiqadda "Paroxetine"? Tilmaamaha loogu isticmaalo dhigayaa in diyaarinta this waxaa maamula si taxadir leh in bukaanka qaba failure beerka, gulukooma xagal-xidho, kelyaha, waali, kelyaha Prostatic benign, dalalka convulsive, xanuunada wadnaha, qalalka. Intaa waxaa dheer, isticmaalka waafaqsan daawada aan waxba ka jirin oo artafiishal, iyo sidoo kale daawooyinka kordhiya halista ah ee dhiig-bax. Waa in aan fiiro gaar ah si ay goobjoog ka ahaayeen sababaha halista cudurada dhiig iyo sahla dalalka cudurka sida.

Niyad jabka "Paroxetine": sida loo qaato daawada?

Waxaan ka fiirsaneysa inay daawada waxaa afka laga qaataa hal mar maalintii (subaxdii) inta lagu jiro quraacda. Kiniiniga in la wada liqo, hoos u maydhay biyo cad.

Inta lagu guda jiro saddexda toddobaad ee ugu horreeya ka dib bilowga daweynta qiyaasta la beddelo si gaar ah. Waxaa markii danbe beddelo (haddii loo baahdo).

Inta lagu jiro murugada qadarka lagu taliyey dheer medicament waa 20 mg maalintii hal mar. Haddii loo baahdo, ee qiyaasta waxaa si tartiib ah kor u kacay 10 mg. Max helay daroogada waa in aanay ka badnaan 50 mg.

Waayo, disorder khasban dose hore waswaaska ee lidka diiqadda ah waa 20 mg maalintii. Intaas ka dib, u kordhiyaa ilaa 10 mg. Qiyaasta talinayaa celcelis ahaan maalin kasta weecasho noocan oo kale ah waa 40 mg. In lagama maarmaan ba'an waxaa lagu kordhin karaa ilaa 60 mg.

Haddii bukaanka uu qabo cudur argagaxa, markii hore ilaa aad qaadi karto ilaa 10 mg ah ee daawada maalin kasta. Si loo yareeyo khatarta suurto galka ah ee Astaamaha argagaxa in qiyaas xiga ee daroogada waxaa kordhay 10 mg. Celcelis ahaan, marka weecasho noocan oo kale ah waa la aqbali karo in la isticmaalo 40 mg "paroxetine" saacadaha, tirada ugu badan - 50 mg.

Marka cuqdadeedka bulshada ama walaaca bulshada xanuunada mugga hore medicament waa in aanay ka badnaan 20 mg maalintii. Haddii daaweynta noocan oo kale ah ka dib markii tarin aan la gaarin, ka dibna 2 todobaad qiyaasta waxaa si tartiib ah kor u kacay in ugu badnaan, in uu yahay ilaa 50 mg maalintii.

In ciladda wallaaca guud daweynta iyo mugga hore ee medicament waa 20 mg maalintii

Haddii bukaanka qaba cudurka beerka ama kelyaha, qiyaasta lagu taliyey waa in ay ahaataa 20 mg maalintii.

dadka waayeelka ah maalin waa la wada baabbi'in karaan wax ka badan 40 mg ah ee daawada.

Si looga hortago astaamaha u-barashada joojin qaadashada daawada waxaa lagu talinayaa in si tartiib tartiib ah.

xaaladood oo badinta

Ma jiraan kiisas ah qiyaasta xad dhaafka la murugada sida "Paroxetine", "Fluoxetine"? Khubarada la ogaado in isticmaalka tiro badan oo ah kaniiniga ay dhab ahaantii si xun u saameyn jidhka bini'aadamka. The lallabo bukaan-aragnimo, afka oo qalala, tachycardia sanka, matag, gariir, gariirka, bradycardia, mydriasis, caro, caro, dhidid, nystagmus, kordhay cadaadiska dhiigga, somnolence, iyo laxanka patrilineal.

Mararka si caddaalad ah u dhif ah, halka la isticmaalayo daroogada daawooyin kale psychotropic, iyo khamriga Suuxdinta waxaa laga yaabaa in bukaan-socodka iyo kala duwanaansho ah ee tilmaan ku saabsan ECG. In xad dhaafka ah u daran, bukaanka waa serotonin syndrome iyo rhabdomyolysis.

Waxa la sameeyo xaaladahan oo kale? In the case of badinta daroogada "Paroxetine" waa in ay ahaataa lavage gastric, oo waxay qaadan doonaan carbon ka shaqeysiin. Haddii loo baahdo, daaweynta calaamadaha.

waxyeellooyin

Waa maxay saamaynta dhinaca daawada keeni kartaa "Paroxetine"? Reviews dhakhtarrada ayaa sheegaya in qalab this runtii waxay ka caawisaa si ay u horumariyaan dhibaato. Kuwaas waxaa ka mid ah xaaladaha iyo cudurada soo socda:

  • On qayb ka mid ah habdhiska dhexe iyo habdhiska durugsan: waali, hurdo, wareer, gariirka, serotonin syndrome, daal, dhalanteed, hurdo la'aan, isku yaacsanaan, madax wareer, udagaashaa, daal, weerarada argagaxa leh, qallal, kacsanaan, xusuus la'aan, jirro extrapyramidal, myoclonus, walwalka.
  • nidaamka muruqyada, tabar-dari muruq, arthralgia, myopathy iyo myalgia.
  • Dareenka: arag isku darsan iyo isku darsamay oo dhan.
  • nidaamka Urinary: kaadida ama haynta kaadida.
  • mareenka dheefshiidka: kordhay ama rabitaanka cuntada, hepatitis, isbedel dhadhanka, afka oo qalala, lalabo, shuban, matag, calool-iyo hoos.
  • nidaamka Taranka: anorgasmia, cillad xagga galmada, hyperprolactinemia ama galactorrhea, kacsi la'aanta iyo xanuunada biyo bax.
  • nidaamka Wadnaha: hypotension orthostatic.
  • Xasaasiyadda: cuncun, finan, anjioedema, iyo urtikaria, ecchymosis.
  • kala duwanaansho kale: rhinitt, dhidid, dheecaan aan habboonayn ee hormoonka antidiuretic, hyponatremia.

Dhexgalka siyaabo kale oo caafimaad

Isticmaalka isku mar ah laabjeexa wax saameyn ah kuma koobin pharmacokinetic iyo nuugista daawada "Paroxetine" ah.

Ahaan uu si loogu isticmaalo hal mar ah lacag na hor leh MAO.

medicament dhaweynta wadajira "paroxetine" daawooyin in la xakameeyo ensaymes beerka, wuxuu u baahan yahay ee loo cayimay marka ugu horeeysa.

cimrigiinnu ku lidka diiqadda dhiig ku saabsan asalka ah ee loo isticmaalo hal mar "ee warfarin."

isticmaalka wadajira ee medicament "paroxetine" la murugada tricyclic, aspirin, neuroleptics atypical, NSAIDs iyo waxay ka dhigan tahay taxane phenothiazine kor nidaamka xinjirowga dhiigga.

Maamulka isku mar la wakiilada serotonergic (sida "tramadol" iyo "sumatriptan") si fudud u keeni kartaa in saamaynta serotonergic wanaajiyey.

Waxaa muhiim ah in la xusuusto!

Si looga fogaado horumarinta syndrome a neuroleptic (malignant), daroogada si taxadar leh u daran "Paroxetine" qoray in bukaanka qaadanayso jirada dhimirka.

dadka waayeelka ah ku saabsan asalka ah ee daroogada waxaa laga yaabaa in hyponatremia.

Marka calaamadaha ugu horeeya ee qalal iyo daaweynta niyad jabka waali la joojiyo.

Inta lagu guda jiro toddobaadyada ugu horeeya ee daaweynta "paroxetine" waxay u baahan tahay la socodka taxaddar bukaanka ay sabab u tahay ismiidaamin ah ay suurto gal.

Inta lagu guda jiro daawaynta waa ka fogaadaan cabitaanka khamriga ay sabab u tahay in ay saamayn sun wanaajiyey.

isticmaalka Carruurta

Drug "Paroxetine" aan qoray in carruurta, sida ay nabadgelyada iyo waxtarka daawaynta bukaanka ee group this aan la aasaasay.

Niyad jabka "Paroxetine": dhigooda

Daawada waxaa lagu beddeli karaa by "Paroxetine"? Waa in la ogaadaa in dawadan, waxaa jira xad ah dhigooda yar. iyaga ka mid ah, waxay noqon lahayd suurad wacan si loo muujiyo daawooyinka soo socda: "Reksetin", "Adepress", "Pliz", "NUSOJ-Paroxetine", "Aktaparoksetin", "Paxil", "sertraline", paroxetine hemihydrat hydrochloride, "" Sirestill "iyo wixii la mid ah.

Si aad u iibsato dhammaan daawooyinka, kuwaas oo farmashiyaha, aad awoodo kaliya by qoro.

Reviews of medicament

Drug "Paroxetine" leedahay wax badan oo ka mid ah dib u eegista isku qasan, labadaba ka xirfadlayaasha iyo bukaanka. Dhinaca mid, waxaa la Mahdiyo waxa ay gacan ka geysaneysaa in xididada loo deg deg ah oo nooc kasta oo niyad-jabka (oo ay ku jiraan qoomiyadda daran, Waxyeelo, oo waxaa la socda walaaca), iyo sidoo kale argagax, waswaaska, guud ahaan iyo bulsho-anxiety disorder. Oo dhinaca kale ah - bukaanno badan ay sheegayaan in isla markiiba ka dib daroogada ay horumariyaan ilaa xad tiro badan oo ah dhibaato. Sidaas darteed, qof ayaa xitaa lahaa in ay joojiyaan daaweynta.

Guud ahaan, khubaro ogow in "Paroxetine" - tani waa daroogada aad wax ku ool ah oo hufan u asiibi karo hawsha loo xilsaaray in ay. Si kastaba ha ahaatee, waxa loo isticmaali karaa oo kaliya ay ku takhasusay ujeedada looga danleeyahay.

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