CaafimaadkaDiyaarinta

"Levocetirizine": tilmaamaha loo isticmaalo, sharaxaad ku saabsan daroogada, analogues iyo dib u eegis

Waa imisa daroogada ah "levocetirizine"? Qiimaha daroogada waxaa loo soo bandhigi doonaa dhamaadka. Waxa kale oo aad baran doontaa sida loo isticmaalo daroogada, ayaa sheegay in uu ka hadlay dhakhaatiirta iyo bukaanka, foomka kuwaas oo waxaa suuq iyo waxa guryaha.

Foomka iyo Halabuurka daroogada Baakadaha

Diyaarinta "Levocetirizine Teva" waxaa soo saaray qaab kiniin. Xoolahooda firfircoon waa dihydrochloride levocetirizine. Sidoo kale daroogada yihiin qaybaha yar ee foomka of laktosmonohydrat lactose, cellulose mikrokristallin, milmahayn magnesium iyo silica Kolloidol.

Iibso medicament tani waxay noqon kartaa in kartoonada, oo waxaa la geeyaa finan aluminium si 7, 14 ama 10 kiniin.

pharmacodynamics daroogada

Maxay yihiin kaniiniyada "levocetirizine"? Tilmaamaha loogu isticmaalo dhigayaa in maalkoodana firfircoon waa isomer levorotatory of cetirizine, kaas oo u dhaqmo sida antagonist aad u xushay oo awood of durugsan H1-receptor.

daroogada viewed saamayn ku yeelan karaan dareen diidmo oo xasaasiyadeed wajiga gistaminozavisimuyu, si loo yareeyo tahriibka ee eosinophils, hoos u permeability vascular iyo sii daayo dhexdhexaadiyayaasha bararka.

Tani ma aha oo kaliya ka hortagtaa horumarinta medicament laakiin sidoo kale attenuates baxsiga ah dareen diidmo oo xasaasiyadeed. Waxa uu ku antipruritic iyo anti-exudative oo uu leeyahay anticholinergic yar iyo saamaynta antiserotoninovoe. Marka qaadasho ku daweyn of daroogada this talinayaa dhow yahay ma keenaan hurdo iyo feejignaan xumo.

Pharmacokinetics

Maxaa xuduudaheedu ogeed leeyihiin "levocetirizine" kiniin? Tilmaamaha loogu isticmaalo ayaa sheegay in ka dib markii dhoos keli ah daawada ay oggolyahay daweynta in 50% bukaannada arkay 12-13 daqiiqo ka dib iyo in 95% bukaanada - ka dib 60 daqiiqo (saamaynta sii inta lagu guda jiro maalmaha xiga).

medicament waxa uu leeyahay pharmacokinetics toosan. Haddii uu qofku cuno waxa ay si degdeg ah u nuugo eegin cunto qaadashada.

bioavailability ee daroogada gaadho 100%. tirada ugu badan ee wakiilka firfircoon arkay 55 daqiiqo ka dib markii uu qofku cuno ka dib, iyo protein qabanaya waa qiyaastii 90%.

Dheef-Drug dhacdaa beerka iyo waxa saxarrada kelyaha in ay ahaanteed.

Tilmaamayaasha

"Levocetirizine" Kiniinka waxa lagu tilmaamayaa lagu daweeyo calaamadaha ka mid ah cudurada soo socda:

  • pollinosis (ama wax-u sanboorka);
  • rhinitt iyo conjunctivitis asal ahaan xasaasiyad, Ulasocto cuncun, lacrimation, rhinorrhea, hindhiso, iyo casaan ah conjunctiva ah;
  • anjioedema,
  • urtikaria, oo ay ku jiraan idiopathic, oo qulqula foomka chronic;
  • dermatosis xasaasiyad, oo waxaa lagu gartaa cuncun iyo finan.

sababo

Waa maxay nooca sababo la ogaado waa in ka hor inta la isticmaalayo "levocetirizine" kiniin? Tilmaamaha loogu isticmaalo Sida laga soo xigtay kuwaas oo laga reebay, sida:

  • da'da ilmaha ilaa lix sannadood ah;
  • CRF noqon daran;
  • inta aad uurka leedahay,
  • diidmo in xubno daroogada, oo ay fiiriyaan in piperazine iyo taagayo daayee;
  • inta lagu jiro naas-nuujinta.

Iyada oo daryeel weyn medicament la qoray noocyada darnaanta fudud iyo kuwa dhexdhexaadka CRF, iyo sidoo kale in da 'weyn (sabab u tahay hoos u suurto gal ah in sifeynta glomerular).

Drug "levocetirizine": tilmaamaha loo isticmaalo

Sida ay tahay, medicament firfircoon ee maamulka afka, iyadoo aan loo eegin isticmaalka cuntada. Kiniinnada waa in la qaato biyo saafi.

Carruurta ka weyn yahay lix sano, sidoo kale bukaanada qaangaarka talinayaa dose hal mar waa 5 mg. Tani waa qiyaasta ugu badan ee maalin kasta.

celceliska muddada daawaynta waa 3-6 toddobaad, iyada oo ku xiran darnaanta calaamadaha. In gaadhista kooban daaweynta xasaasiyadda in la buuxiyaa karaa hal toddobaad gudahiisa.

Sida xaaladaha raaga, xasaasiyad, waxay u baahan karaan daroogada muddo lix bilood ah.

bukaanada waayeelka ah iyo kuwa qaba cudurka beerka uma baahnid inaad qabsato qiyaasta.

Marka qiyaasta cudur kalyaha ah in la waafajiyo sida ay QC bukaanka:

  • ka yar 10 ml halkii daqiiqo - qaata dawooyinka u wanaagsanayn;
  • ka yar 30 ml halkii daqiiqo - 5 mg 6 maalmood oo dhan;
  • 30-49 ml halkii daqiiqo - 5 mg of 4 maalmood oo dhan;
  • in ka badan 50 ml halkii daqiiqo - 5 mg 2 maalmood.

dhibaato

Waa maxay dhibka uu dhici kara inta aad qaadanaysid kaniiniga "levocetirizine"? khubaro Guest ayaa sheegaya in dhibaato soo socda:

  • daal, madax xanuun, wareer, xanaaq,
  • hurdo, aragga indhaha oo isku darsamay, calool xanuun, madax xanuun,
  • dareen ah qallayl ee afka, dyspepsia, dyspnea, daal ah,
  • lalabo, miisaanka oo kordha, tachycardia;
  • cadaanyo sida anjioedema, finan maqaarka, cuncun, urtikaria ee.

Calaamadaha badinta

Marka la helo in ka badan hal kiniin maalin kasta in bukaanada qaangaarka ah u horumariyaan hurdo, iyo carruurta - reyn iyo walwalka.

therapy ee xaaladaha sida waa la dhimay si Calaamadaha lavage iyo qaadashada sorbents gastric.

isdhexgalka daroogada

soo dhaweynta wadajira "levocetirizine" with "theophylline" at dose oo ah 400 mg, yaraynaysaa ansixin guud ee 16% ugu horeysay, laakiin ma bedeli ku kinetics doonana.

In dadka xasaasi ah wada-maamulka daroogada la wakiilada in la xakameeyo habka dhexe ee neerfayaasha, oo ay ku jiraan ethanol, potentiate karaan dhibaatooyinka soo dampening.

Micne ah, analogs, iyo kharashka daawada

Waa maxay analogues daroogada "levocetirizine" ah? Dhibcood ee maamulka afka ku yeelan kartaa saameyn la mid ah sida kiniin ah. Sidaa darteed, khubarada qaar ka mid ah ku talinaynaa beddelayo hab sida daroogada loo tixgeliyaa sida "Pollezin" iyo "Suprastineks" (dhibcood). Intaa waxaa dheer, analogs daroogada this waa "Allertsetin ',' Zestril ',' Alerza", "Rolinoz", "Zirtek", "Zintset", "Tsetrin", "Allertek", "Zetrinal", "Amertil" "cetirizine" "Zodak", "Letizen S", "Parlazin".

Sida micne ah, ka dibna si daawooyin sida waxaa ka mid ah kuwan soo socda: "Zodak" Allerset-L "," Zenaro "," levocetirizine "Sandoz", "Tsetrilev", "ee L-CET", "Tsezera", "Glentset", "Suprastineks" "Aleron" Express "," Ksizal ".

ma daroogada this sida "levocetirizine" Intee in leeg? Its qiimaha kala duwan yihiin inta u dhaxaysa 170-290 rubles.

Kurtumm

Inta badan dib u eegista ku saabsan daroogada "Levocetirizine-Teva" fiican. bukaan badan oo si joogto ah ay dhibaatadu ka kiciyaan cadaanyo kala duwan, marar aad u isticmaalaan daroogada this. Waxay ku doodayaan in "levocetirizine" waa qalab wax ku ool ah oo keliya ma aha, waayo, therapy muddo dheer, laakiin sidoo kale gargaarka degdegga ah haddii ay dhacdo of xasaasiyad xilliyeed ama sanadka oo dhan. diyaarinta wuxuu kuu ogolaanayaa inaad si ay u ilaaliyaan caafimaadka heerka ugu habboon, baabi'inta dhammaan calaamadaha xun ee nooca xasaasiyadda.

Ka mid ah dib u eegista xun waxaad ka heli kartaa kuwa kaas oo nidhaahno, daroogada sababa hurdo, daal iyo caro. Dhakhaatiirta ayaa sheegay in in marka la helo qiyaasta saxda ah ee daawada falcelin ku qoran tahay mid aad u dhif ah.

"Levocetirizine" ama "Cetirizine", taas oo ka wanaagsan?

Su'aashani waxay la waydiiyo by bukaanno badan oo si joogto ah ay dhibaatadu ka dareen diidmo oo xasaasiyadeed. Khubarada sheegaan in labada bandhigay daroogada ku ool ah ay ula qabsadaan hawsha. Laakiin, sida dhaqanka shows, "levocetirizine" cover kiniin iyo meesha tiro badan oo ah calaamadaha xasaasiyad.

Mid ka mid ah ma dhihi karo in "cetirizine" Waxa jira noocyo dhowr ah oo loo sii daayo (dhibciyo, kiniin, sharoobo). Taasina waxay keentaa in ay ka badan habboon in la isticmaalo, gaar ahaan carruurta (lix sanno).

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