CaafimaadkaDiyaarinta

"Betacam": tilmaamaha loo isticmaalo, analogs iyo dib u eegis

Si aad u baabi'iyo cadaadiska sare iyo cudurada wadnaha kala duwan iyadoo la isticmaalayo hab adrenoblokatornye beta1. Mid ka mid ah daawada sida waa daroogada ah "Betacam". Tilmaamaha loogu isticmaalo qeexayaa isaga sida daroogada in soo bandhigaa cardioselective, antihypertensive iyo sympathomimetic tallaabo.

Calaamadaha caadiga ah

Tani waxaa loo arkaa qalab dardaro beta1-adrenergic xanibaha. Soo saaray warshad Cyprus "Medokemi LTD" kiniin la galkeeda cad ama si xooga cad daahan.

Drug "Betacam" edbinta ku saabsan sharaxaad ka mid ah daroogada ee ku jira qof soo socda: waxay u sameeyaan a meelaha lenticular fekrado, waxaa jira aaladda wax kala qaybinaysa qaab halis ah. Haddii aad jebiso kiniin ah oo kasta, ka dibna waxa ay noqon doontaa waxyaabaha ku cad gudaha ama ku dhowaad caddaan.

On medicament "Betacam" edbinta on description xirmo macaamilka soo bandhigaysaa sida soo socota: hal pack ka kooban yahay saddex finan. Mid kasta oo saxanka gacanta dusha waxaa soo baakadeeyey at 10 kiniin.

Qaab-dhismeedka

In daawada doorka ugu weyn waxaa la siiyaa qayb hadda qaab cusbo hydrochloride betaxolol. qiyaasta The oo kiniin kasta waa 0,020 g

hab A of "Betacam" edbinta ee curinta waxay maaddooyinka firfircoonayn tilmaamay aan la tilmaamayo tiradoodu. Kiniiniga sameeyay glycolate starchy sodium, sonkor, caano, milmahayn magnesium, mikrokristallin nooca cellulose, aerosil, xabagta titanium, iyo tones polyetylen hydroxymethylpropylcellulose sumadda 400.

hab of action

On daawo "Betacam" diiwaanka Xaqiijiyay beta1 cardioselective -adrenoblokatornuyu aan saamayn waxqabad sympathomimetic kala go'lahayn. Oo looxyadu waxay muujiyaan xuub xasilinta waxtarka saboolka ah.

dhaqdhaqaaqa Antihypertensive waxaa sabab u ah falalka in la yareeyo wax soo saarka ee wadnaha ee muruqa wadnaha iyo in la yareeyo kicinta dabacsanaadaan in xididdada dhiigga ee ubucda ah.

saamaynta Selectivity daroogada on formation of β 1 -adrenoreceptor ma la odhan karaa shuruud la'aan, sababtoo ah qaadasho sare ee betaxolol saamayn ku yeelan kara β formation -adrenozavisimye 2 receptor kaasoo ku yaala weelashii hawomareenno iyo dhiig.

Joojinta tallaabada of daroogada, iyada oo la tixgelinayo sifooyinka pharmacodynamic la xidhiidha hoos u dhac in garaaca wadnaha waqtiga nasashada iyo waqtiga layliga. Waxaa sabab u ah Iscelin ee qaababka β-adrenoceptor in Guntin Dalqada wadnaha, taas oo yaraysa ay automaticity.

Waxa kale oo ay yaraynaysaa sii daayo myocardial cajiib ah in xaalad firfircoon oo dadban ee jirka, oo ka dhalata iska soo horjeeda ee tartan rasmi ah ee catecholamines iyo dhammaato dareemayaasha durugsan nooca adrenergic.

Daawada yaraynaysaa cadaadiska dhiigga systolic iyo diastolic halbowleyaasha waqtiga nasashada iyo waqtiga jimicsiga, yaraynaysaa kordhay orthostatic reflex in inta jeer ee foosha wadnaha. Noocan oo kale ah saamayn of daroogada yaraynaysaa load ku on myocardium ah.

Beta adrenoblokatornoe daawaynta ayaa antihypertensive hawlaha by soo socda hab:

  • hoos u wax soo saarka wadnaha;
  • hareen dabac ku dhaca halbowle ee maqnaadaan sabab u tahay tallaabo dhexe, kaas oo xaddidaya wadnaha u dabacsanaadaan derbiyada vascular inta lagu guda jiro ku istaago hawl renin.

Maamulka muddada dheer ee daroogada ma yareeyo saamaynta ay hypertensive. Haddii aan qaato dhoos keli betaxolol 0,005 ama 0.04 g, hoos u cadaadiska muujin doonaa 3 kaliya ka dib ama 4 saac.

In daawada, "Betacam" Codsiga User waxay muujinaysaa in maamulka a 0.005g qiyaasta sababta saamayn antihypertensive kuwaas oo xoogooda waa laba jeer ka hooseeya iyadoo kiniin oo dhan.

hawlaha ugu badan antihypertensive fiirsashada wax ka mid ah betaxolol muuqataa 7-14 maalmood ka dib.

qiyaasta daweynta daawo ma keeno saamayn cardiodepressivny fahmayaan, saameyn ah kuma laha dheef glucose, hana u kordhinnin dib u dhac ah ee siifilisku sodium iyo dheecaanka in unugyo ka.

Maxaa loo isticmaalaa

Drug "Betacam" edbinta sanduuqa markhaatiga kor saaran waxaa ka mid ah khadadka soo socda:

  • cadaadiska dhiigga ee sareeya,
  • cudurka halbowlaha wadnaha muruqyada cajiib ah myocardial, Wadnaxanuun myocardium in geeddi-socodka;
  • cardiomyopathy hypertrophic.

Dawada waxa qoray marka ay jiraan isbedel ee wadnaha, kuwaas oo muujiyay in xawaaraha ee laxanka sanka, tachyarrhythmias ventricular iyo dabeecadda supraventricular, dib u depolarization ee myocardium ah, arrhythmia la xidhiidha prolapse ee waalka mitral, wax soo saarka-dhaafka ah ee hormoonnada thyroid.

Sida loo isticmaalo

On daawo tilmaamaha "Betacam" for isticmaalka rinjiga qiyaas ku xiran xaaladda bukaanka. All maalin dose cabniinka per la cabbo. Cuntada wax saameyn ah kuma nuugista daawada. kaniini waa in la hoos u maydhay biyo nadiif ah.

La kordhiyo cadaadiska dhiigga loola dhaqmo dose bilaabo maalin kasta ee ka 0,005 in 0,010 g Ka dib 7 ama 14 maalmood, haddii loo baahdo, in la kordhiyo xaddiga medicament 0,020 g

Waa in aan isticmaalo

Ma aha qof kasta oo u ogolaanaya isticmaalka hab ah "Betacam" diiwaanka. Sababo la xiriira la-dhaafka ah u nuglaan ah maaddooyinka, iyo sidoo kale betaxolol hydrochloride.

Waxaa la ma qoro ee bukaanada qaba muruqa wadnaha chronic foomamka la'aan sinoatrialnuyu iyo xannibaad atrioventricular in darajadii labaad, iyo kii saddexaad, bradycardia, hypotension, weeraro neef bronki, angina lama filaan ah.

Daawooyinka "Betacam" tilmaamaha pill loo isticmaalo waxaa sidoo kale aan lagu talinayaa in iyada iyo alaabtan oo dhamaadka angiotrofonevroze nooca lama filaan ah cardiogenic cabbaan, sii kordhaya muruqyada cajiib ah myocardial, ophthalmoplegia asthenic, endarteritis obliterans, lesions emfizemnom unugyada sambabada, obstructive nooca boronkiitada mellitus diabetes chronic.

isbedel cad in kelyaha iyo lesions psoriatic waa u ah oo lagu daweeyo.

dhibaato

waxyeello ka soo gaartey waxay ka dhigan tahay "Betacam" codsiyada User waxaa ka mid ah garaaca wadnaha gaabis ah, xannibaad atrioventricular, la'aan muruqyada wadnaha, hoos u orthostatic in cadaadis, wareegga dhiigga oo xun agagaarka maqnaadaan, gacmaha inta badan iyo lugo qabow, paresthesia. Sidaas carqaladeeyey nidaamka vascular iyo waxyaalaha qalbiga ku jira.

dabac bronki, finan, urtikaria, psoriasis, isha qalalan xuubdheecaanka dhici kara dareen diidmo oo dhinac ah iyo xubnaha muuqaal ah neefsashada, maqaarka.

daroogada waxay keeni kartaa hurdo, xaalad asthenic, xanuunada niyad, daal xad-dhaaf ah, wareer, calaamadaha dhalanteed, xanuun wareer iyo madax xanuun.

hababka loo baahnayn ee habka dheef shiidka xiriirka la leh lallabo, retching, shuban, cholestasis kursiga dib u dhac.

daliilka kale garoomada daroogada uma shaqayn karo sidii hoos u dhac in leukocyte iyo unugyada dhiigga xinjirowga, iyo sidoo kale awoodba dhimay.

Features ee daaweynta

Aqbalaada daroogo kasta la xidhiidha laga yaabaa in la Gudigga gaar ah, taas oo ku xiran kooxaha pharmacological, ka kooban oo qiyaasta of daroogada loo isticmaalo.

Daawooyinka "Betacam" edbinta ku saabsan isticmaalka tilmaamaha gaarka ah waxaa la siiyaa waayo, kiis kasta oo ka mid ah non-caadiga ah, oo u baahan fiiro gaar ah.

Sidaas daraaddeed markii hore stage of daaweyn may sabab la'aan wadnaha muruqa in dadka nugul this weecasho.

Kiniinka "Betacam" waji calaamadaha a hypoglycemic gobolka, inta badan kaas oo waxaa loo arkaa a xadgudub ku ah wadnaha laxanka. Tani waa in ay qaadaan aqoonta akoonka bukaanka qaba kacsantahay dhiig sonkorta. Waxay u baahan tahay la socodka joogtada ah ee heerka sonkorta dhiigga.

Haddii aad isticmaasho dawooyinka, buuga "Betacam" (kiniin) edbinta ku talinaysaa lacag bixisid si aad gacanta ugu garaaca wadnaha dareenka. In case of cudurada laxanka sanka bradycardic, qiyaasta loo baahan yahay si loo yareeyo ama burin wakiilka daaweynta xogta.

Waxay u baahan tahay isticmaalka taxadir daroogada ee bukaanka qaba waxbarashada pheochromocytoma.

Isku daroogada miisaaniyadda in la qabtaa suuxdinta neefsasho, sababa Iscelin of shaqo cajiib ah myocardial muruqyada iyo yareynta dhiig-karka. Non-depolarizing dabcineyso muruqa muujiyaan a kiniiniyada tallaabo dheer degganayn markii loo feydo "Betacam".

Haddii aad rabto in aad si ay u fuliyaan dabeecad qorsheeyey qalliinka-gelinta, diyaarinta baajiso laba maalmood ka hor ay dhacdo in Alwaaxdii ma saamayn suuxinta guud.

Daawada si ay u joojiyaan daaweynta tilmaamaha "Betacam" si loogu isticmaalo ma taliyaa mar, laakiin wareega, iyadoo hoos u dhac ku kacmaha 7 ama 14 maalmood, si looga fogaado dareen-celin jirka ee in la baabiiyo of daroogada. saddex maalmood oo kasta xaddiga daroogada waa la dhimay by 0,005 g

Kiniiniga aan la qaadan daawooyinka in ay yihiin retarders enzyme oxidase Monoamine.

saamaynta Hypotensive daroogada iyo in la yareeyo daawooyinka anti-estrogen magnyl in dib u udhigo sodium iyo biyo, iyo sidoo kale la xakameeyo ereygu wuxuu ahaa ee xeryahooda prostaglandin gudahood kelyaha.

isticmaalka wadajira ee diltiazem, verapamil iyo kiniiniyada amiodarone leh "Betacam" keenaysaa in kordhay tallaabo inhibitory of hydrochloride betaxolol on contractility ee myocardial cajiib ah murqaha iyo tabinta.

The isku darka daawada la wadnaha glycosidic daroogada kor u atrioventricular block nooca.

Isku dhafan oo antihypertensives kale waxay kordhisaa kiniin hawl hypotensive "Betacam".

Cocaine hoos u oggolyahay ku daweyn of betaxolol ay maamulka isku mar.

isku darka ah "Betacam" kiniin agonister ama xanthines sababa daciifisa labada dhinac ka mid ah waxqabadka.

Phenothiazines iyo betaxolol hydrochloride by ficil kordhin ay ka kooban tahay ee dhiigga.

Daawo "Betacam" hortagtaa diyaar u qaadidda ka kooban lidocaine ama theophylline.

Sulfasalazine korodhka serum fiirsashada of betaxolol hydrochloride.

Ma jiro macluumaad ku saabsan isticmaalka daroogada ee dadka bukaanka ah ee carruurnimada.

Digniin loo baahan yahay in codsiga ah ee kiniiniyada in dadka halka baabuur-wadidda baabuurta ah, iyo sidoo kale dumarka uurka leh iyo kuwa nuujinaya.

qalabka

By beta1-adrenoblokatornym Drug Administration u soocay daawo "Betacam" barashada buuga. Analogs sidoo kale waxay ka tirsan yihiin class this of pharmacotherapeutic. Waxay ka kooban falimihiisii kale qayb firfircoon sida hydrochloride betaxolol.

Faransiis waxaa loo arkaa ah analog oo ka mid ah daroogada "Lokren", soo saaray "Sanofi Winthrop Industry" ee foomka of a kiniin dahaarle cad film. Form iyaga ku wareegsan oo la biconvex wejigooda, taas oo halis yaalo iyo kala gadaaman naqshada "ke 20".

Waxaa jira dhoos keli ah 0.02 g of hydrochloride betaxolol. daawo qaybaha darran waxaa ka mid ah sonkorta caanaha, cellulose mikrokristallin, carboxymethyl sodium nooca A, Silicon Kolloidol dioxide, milmahayn magnesium.

Halabuurka daahan filim ayaa lagu ogaan karaa hypromellose, polyetylen tones sumadda 400, titanium dioxide.

Daroogada lagu iibiyo baakad baakadaha la laba finan of 14 kiniin.

daawo si loo baabi'iyo cadaadis dhiig oo sareeya codsatay, waxaa sidoo kale lagu daro daawooyinka kale ee ka dhanka ah hypertension.

Daawada qaadi karaan tallaabooyin ka hortag ah si wax looga qabto sii daridda ah ee angina foom kacsan.

daawaynta la mid Ruush yahay daawo "Betaxolol", kaasoo lagu soo saaro by "Moscow hormoonada jidhka Plant" oo ah qaab kiniin cad dahaarka leh. Waxay leeyihiin qaab wareegsan oo wejigooda biconvex. Walaxda firfircoon waxaa loo arkaa betaxolol hydrochloride qadarkuu of 0,020 g maaddooyinka darran waxaa ka mid ah sonkorta caanaha, istaarijka sodium, ammooniya aerosil, milmahayn magnesium, mikrokristallin nooca cellulose. daahan filim waxaa la aasaasay by khamriga polyvinyl dioxide-titanium, Rusheyn kartaa, Macrogol 3350 brand, Opadry cad-2.

Qalabkan waxaa loo habsami ah loo isticmaalo cadaadis dhiig oo sareeya.

Waxaa jira daawo ah "" Betaxolol "ee foomka of dhibcood isha in lagu dabaqo laga dhayayo in-xagal furan nooca glaucoma chronic, iyadoo cadaadis sare intraocular, soo celinta aragti ka dib markii faragelinta trabekuloplasticheskogo laser.

opinion bukaanka

About macnaheedu yahay "Betacam" tilmaamaha isticmaalka cawaaqib aan loo baahnayn ee dib u eegista waxaa ka mid ah qaybta "Xasaasiyada Dacdarrada". calaamadahan laga yaabaa in aanay daruuri dhacaan marka la isticmaalayo daroogada.

Bukaan badan ayaa laga maqli karaa ra'yi-celin wanaagsan oo ku saabsan beta1-adrenoblokatornom macnaheedu yahay "Betacam" in si fiican oo daawaynaya hypertension iyo angina. Asal ahaan qaadan kiniiniyada wada daawooyin kale antihypertensive in therapy adag in kor loogu qaado waxtarka ay.

daaweynta cadaadiska dhiigga celinta Post si caadi ah, taas oo si weyn u soo hagaagaysa caafimaadka bukaanka.

Waxaa sidoo kale jira dib u eegista ah ee daroogada in ay muujiyaan waxtardarradoodu daaweynta wakiilka this.

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